SCHEMBL5583408

SCHEMBL5583408

Fc1cc2c(c(-c3cccnc3)c1)O[CH]C2

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 4/20 0.42
TDO2 P48775 3/20 0.40
CYP11B1 P15538 8/20 0.39
CYP11B2 P19099 7/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.38
NPY5R Q15761 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP2A6 P11509 1/20 0.38
GPR84 Q9NQS5 1/20 0.37
PDE4B Q07343 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27723763 0.83 NPC1 (0.42) CYP11B1CYP11B2CYP1A2NPY5RCYP2A6
SCHEMBL5583665 0.80 CYP11B1 (0.47) CYP17A1TDO2CYP11B1CYP11B2CYP1A2
SCHEMBL27723761 0.77 PTGS2 (0.35) TDO2CYP11B2CYP3A4ALDH1A1GPR84
SCHEMBL4597056 0.75 TDO2 (0.38) CYP17A1TDO2CYP11B1CYP11B2CYP1A2
SCHEMBL4597059 0.75 PARP1 (0.47) CYP17A1TDO2CYP11B1CYP11B2CYP1A2
SCHEMBL27723664 0.74 AQP1 (0.36) GPR84
SCHEMBL27723675 0.73 KDM1A (0.41) TDO2CYP1A2CYP3A4NPY5RALDH1A1
SCHEMBL4224624 0.72 AQP1 (0.55) CYP17A1TDO2CYP11B1CYP11B2CYP1A2
SCHEMBL27703115 0.70 MAPT (0.39) GPR84
SCHEMBL27723658 0.70 TAAR1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101448492-A Methods of treating cognitive and other disorders WYETH CORP (US) 2009-06-03 CN claimed
CN-101389325-A Treatment of drug abuse WYETH CORP (US) 2009-03-18 CN claimed
CN-101203217-A Methods for modulating bladder function WYETH CORP (US) 2008-06-18 CN claimed
CN-101198323-A Therapeutic combinations for the treatment or prevention of psychotic disorders WYETH CORP (US) 2008-06-11 CN claimed
CN-101198322-A Novel therapeutic combinations for the treatment or prevention of depression WYETH CORP (US) 2008-06-11 CN claimed
CN-101189004-A Treatment of pain WYETH CORP (US) 2008-05-28 CN claimed
JP-2007509174-A 2007-04-12 JP claimed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP claimed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO claimed
CN-101448492-A Methods of treating cognitive and other disorders WYETH CORP (US) 2009-06-03 CN disclosed
CN-101389325-A Treatment of drug abuse WYETH CORP (US) 2009-03-18 CN disclosed
CN-101203217-A Methods for modulating bladder function WYETH CORP (US) 2008-06-18 CN disclosed
CN-101198323-A Therapeutic combinations for the treatment or prevention of psychotic disorders WYETH CORP (US) 2008-06-11 CN disclosed
CN-101198322-A Novel therapeutic combinations for the treatment or prevention of depression WYETH CORP (US) 2008-06-11 CN disclosed
CN-101189004-A Treatment of pain WYETH CORP (US) 2008-05-28 CN disclosed