SCHEMBL5586175

SCHEMBL5586175

O=CCCC(I)c1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.32
TDO2 P48775 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC11 Q96DB2 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
HDAC9 Q9UKV0 1/20 0.32
HDAC5 Q9UQL6 1/20 0.32
SLC6A3 Q01959 1/20 0.32
GABBR2 O75899 1/20 0.32
GABBR1 Q9UBS5 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
LOXL2 Q9Y4K0 1/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL67251 0.80 CYP19A1 (0.41) MEN1LMNAKMT2AHTT
SCHEMBL26106019 0.77 IDO1 (0.32) IDO1TDO2HDAC3HDAC4HDAC1
SCHEMBL26109029 0.77 IDO1 (0.32) IDO1TDO2HDAC3HDAC4HDAC1
SCHEMBL6223969 0.77 IDO1 (0.32) IDO1TDO2HDAC3HDAC4HDAC1
SCHEMBL27999842 0.77 HTT (0.37) MEN1LMNAKMT2ASMN1; SMN2HTT
SCHEMBL13619654 0.77 AOC3 (0.44) SLC6A3GABBR2GABBR1MEN1LMNA
SCHEMBL21855589 0.76 CYP19A1 (0.45) MEN1LMNAKMT2ASMN1; SMN2HTT
SCHEMBL6871140 0.74 GABBR2 (0.37) IDO1TDO2HDAC3HDAC4HDAC1
SCHEMBL9047470 0.74 ALDH1A1 (0.40) IDO1TDO2SLC6A3LOXL2MEN1
SCHEMBL3417295 0.74 AOC3 (0.36) IDO1TDO2HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1763523-A1 QUINAZOLINEDIONE DERIVATIVES AS PARP INHIBITORS JANSSEN PHARMACEUTICA N.V. (BE) 2007-03-21 EP disclosed
WO-2006003148-A1 QUINAZOLINEDIONE DERIVATIVES AS PARP INHIBITORS JANSSEN PHARMACEUTICA N.V. (BE) 2006-01-12 WO disclosed