Fumaric Acid

Fumaric Acid

SCHEMBL5586404

O=C(O)C=CC(=O)O.O=C(O)CC(OC(CC(=O)O)C(=O)O)C(=O)O

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ATP4AATP4BAXLBTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CHRM2CHRM3CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4FLT3HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3KCNH2KMT2AMAP2K1MAP2K2MEN1MLNRMPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PLK4PPARGRENS1PR1SLC6A2SLC6A3SLC6A4SMOTYK2atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Fumaric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.41
TP53 P04637 1/20 0.41
EGLN1 Q9GZT9 1/20 0.41
EGLN3 Q9H6Z9 1/20 0.41
TDP1 Q9NUW8 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.37
HCAR2 Q8TDS4 5/20 0.35
SLC22A6 Q4U2R8 1/20 0.35
FOLH1 Q04609 1/20 0.32
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
GABRR1 P24046 2/20 0.31
GABRR2 P28476 2/20 0.31
BLM P54132 2/20 0.31
GABRR3 A8MPY1 1/20 0.31
LMNA P02545 1/20 0.31
APEX1 P27695 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL5586403 1.00 TSHR (0.41) TSHRTP53EGLN1EGLN3TDP1
Malic Acid SCHEMBL9406592 0.90 SMN1; SMN2 (0.56) TSHRTP53EGLN1EGLN3TDP1
SCHEMBL30293 0.88 TDP1 (0.48) TSHRTDP1SMN1; SMN2SLC22A6FOLH1
SCHEMBL8558212 0.85 TDP1 (0.46) TSHRTDP1SMN1; SMN2SLC22A6FOLH1
SCHEMBL9406499 0.85 TDP1 (0.46) TSHRTDP1SMN1; SMN2SLC22A6FOLH1
SCHEMBL9406869 0.85 TDP1 (0.46) TSHRTDP1SMN1; SMN2SLC22A6FOLH1
SCHEMBL9053647 0.85 TDP1 (0.46) TSHRTDP1SMN1; SMN2SLC22A6FOLH1
Ammonia Solution, Strong SCHEMBL28156292 0.85 TDP1 (0.52) TSHRTDP1SMN1; SMN2SLC22A6FOLH1
SCHEMBL646453 0.81 HCAR2 (0.50) TSHRTP53EGLN1EGLN3TDP1
SCHEMBL3716837 0.81 HCAR2 (0.50) TSHRTP53EGLN1EGLN3TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3942011-B2 2007-07-11 JP claimed
EP-1235820-B1 ETHER-CAPPED POLY(OXYALKYLATED) ALCOHOL SURFACTANTS PROCTER & GAMBLE (US) 2006-08-23 EP claimed
US-6844309-B1 Ether-capped poly(oxyalkylated) alcohol surfactants THE PROCTER & GAMBLE COMPANY (US) 2005-01-18 US claimed
JP-2003516424-A 2003-05-13 JP claimed
EP-1235820-A2 ETHER-CAPPED POLY(OXYALKYLATED) ALCOHOL SURFACTANTS THE PROCTER & GAMBLE COMPANY (US) 2002-09-04 EP claimed
WO-2001042408-A2 ETHER-CAPPED POLY(OXYALKYLATED) ALCOHOL SURFACTANTS THE PROCTER & GAMBLE COMPANY (US) 2001-06-14 WO claimed