SCHEMBL5591471

SCHEMBL5591471

CN1CCC(CN2CCN(Cc3ccc(C(=O)NN(CC4CCCC4)c4nc(C#N)ncc4Br)cc3)CC2)CC1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 5/20 0.69
CTSK P43235 5/20 0.69
CTSL P07711 4/20 0.69
CTSB P07858 1/20 0.69
HDAC6 Q9UBN7 1/20 0.39
PRKAA2 P54646 2/20 0.39
TBK1 Q9UHD2 3/20 0.38
IKBKE Q14164 2/20 0.37
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36
KLKB1 P03952 1/20 0.36
KLK1 P06870 1/20 0.36
KIT P10721 1/20 0.35
FLT3 P36888 1/20 0.35
PRKAB2 O43741 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKAA1 Q13131 1/20 0.35
PRKAG3 Q9UGI9 1/20 0.35
PRKAG2 Q9UGJ0 1/20 0.35
PRKAB1 Q9Y478 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5591423 0.95 CTSS (0.76) CTSSCTSKCTSLCTSBHDAC6
Trifluoroacetic Acid SCHEMBL5591828 0.95 CTSS (0.63) CTSSCTSKCTSLCTSBHDAC6
SCHEMBL5591415 0.94 CTSS (0.67) CTSSCTSKCTSLCTSBHDAC6
SCHEMBL5591180 0.93 CTSS (0.68) CTSSCTSKCTSLCTSBHDAC6
SCHEMBL8245361 0.92 CTSS (0.58) CTSSCTSKCTSLCTSBHDAC6
SCHEMBL5591425 0.91 CTSS (0.67) CTSSCTSKCTSLCTSBHDAC6
Trifluoroacetic Acid SCHEMBL5591441 0.91 CTSS (0.69) CTSSCTSKCTSLCTSBHDAC6
SCHEMBL3165989 0.90 CTSS (0.66) CTSSCTSKCTSLCTSBHDAC6
SCHEMBL5591580 0.90 CTSS (0.65) CTSSCTSKCTSLCTSBHDAC6
SCHEMBL5590944 0.90 CTSS (0.68) CTSSCTSKCTSLCTSBHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO claimed
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed