SCHEMBL5591580

SCHEMBL5591580

N#Cc1ncc(Br)c(N(CC2CCCC2)NC(=O)c2ccc(CN3CCN(CCO)CC3)cc2)n1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.65
CTSK P43235 4/20 0.65
CTSL P07711 4/20 0.65
CTSB P07858 1/20 0.65
PRKAA2 P54646 8/20 0.36
HDAC6 Q9UBN7 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC8 Q9BY41 1/20 0.35
PRKAB2 O43741 3/20 0.34
PRKAG1 P54619 3/20 0.34
PRKAA1 Q13131 3/20 0.34
PRKAG3 Q9UGI9 3/20 0.34
PRKAG2 Q9UGJ0 3/20 0.34
PRKAB1 Q9Y478 3/20 0.34
KDM4E B2RXH2 1/20 0.34
TBK1 Q9UHD2 1/20 0.34
HDAC4 P56524 1/20 0.34
KCNH2 Q12809 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5591481 0.95 CTSS (0.60) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL5591425 0.93 CTSS (0.67) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL5591423 0.93 CTSS (0.76) CTSSCTSKCTSLCTSBHDAC6
SCHEMBL5590923 0.92 CTSL (0.60) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL5591422 0.91 CTSL (0.62) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL5591383 0.91 CTSL (0.63) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL5591471 0.90 CTSS (0.69) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL5591415 0.90 CTSS (0.67) CTSSCTSKCTSLCTSBPRKAA2
SCHEMBL5591180 0.89 CTSS (0.68) CTSSCTSKCTSLCTSBHDAC6
Trifluoroacetic Acid SCHEMBL5591489 0.88 CTSS (0.61) CTSSCTSKCTSLCTSBPRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO claimed
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed
WO-2007025774-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed
WO-2007025776-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed