SCHEMBL5592005

SCHEMBL5592005

N#Cc1c(CO)cc(-c2ccccc2)cc1C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.48
ALDH1A1 P00352 6/20 0.48
HPGD P15428 5/20 0.48
GAA P10253 4/20 0.48
GLA P06280 3/20 0.48
L3MBTL1 Q9Y468 4/20 0.45
TDP1 Q9NUW8 2/20 0.45
NPSR1 Q6W5P4 1/20 0.43
AR P10275 6/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
RXRA P19793 3/20 0.40
RXRB P28702 2/20 0.40
RXRG P48443 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
PGR P06401 1/20 0.40
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5592001 0.85 KDM4E (0.48) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL24749451 0.82 KDM4E (0.56) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL25983810 0.78 KDM4E (0.52) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL3906275 0.76 KIF11 (0.49) ARRXRARXRBRXRG
SCHEMBL27863089 0.75 ALDH1A1 (0.40) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL2652120 0.74 KIF11 (0.51) RXRARXRBRXRG
SCHEMBL15534698 0.74 P2RX7 (0.44) NPSR1ARLMNA
SCHEMBL24751432 0.72 AR (0.59) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL25994171 0.70 AR (0.51) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL1373309 0.70 AR (0.58) ARRXRARXRBRXRGPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007121389-A2 4,4-DISUBSTITUTED PIPERIDINE DERIVATIVES AS NK-I AND SEROTONIN TRANSPORTER INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-10-25 WO disclosed