SCHEMBL5592572

SCHEMBL5592572

CC(C)CN(NC(=O)c1ccc(CN2CCN(CCCN3CCCCC3)CC2)cc1)c1nc(C#N)ncc1Cl

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.70
CTSK P43235 4/20 0.70
CTSL P07711 3/20 0.70
CTSB P07858 2/20 0.70
TBK1 Q9UHD2 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
MELK Q14680 1/20 0.37
RAPGEF3 O95398 1/20 0.35
F10 P00742 1/20 0.35
MC4R P32245 3/20 0.35
PTGER1 P34995 1/20 0.35
IKBKE Q14164 1/20 0.35
TNF P01375 1/20 0.35
EGFR P00533 1/20 0.35
HRH3 Q9Y5N1 3/20 0.35
MC5R P33032 1/20 0.35
MC3R P41968 1/20 0.35
MC1R Q01726 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5592915 0.97 CTSS (0.72) CTSSCTSKCTSLCTSBTBK1
SCHEMBL5592755 0.96 CTSS (0.73) CTSSCTSKCTSLCTSBTBK1
SCHEMBL8242433 0.95 CTSL (0.71) CTSSCTSKCTSLCTSBTBK1
Trifluoroacetic Acid SCHEMBL5592680 0.95 CTSS (0.64) CTSSCTSKCTSLCTSBTBK1
SCHEMBL5592866 0.94 CTSL (0.72) CTSSCTSKCTSLCTSBTBK1
SCHEMBL5592751 0.92 CTSL (0.59) CTSSCTSKCTSLCTSBPTGER1
SCHEMBL5592558 0.91 CTSL (0.73) CTSSCTSKCTSLCTSBTBK1
SCHEMBL5592944 0.91 CTSL (0.73) CTSSCTSKCTSLCTSBTBK1
SCHEMBL8243023 0.91 CTSS (0.83) CTSSCTSKCTSLCTSBTBK1
SCHEMBL8243570 0.90 CTSL (0.67) CTSSCTSKCTSLCTSBTBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025775-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed
WO-2007025776-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed