SCHEMBL5595287

SCHEMBL5595287

COC(=O)c1cc(Br)c(N)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.53
ABL1 P00519 1/20 0.51
NQO2 P16083 5/20 0.47
KDM4E B2RXH2 6/20 0.46
ALDH1A1 P00352 5/20 0.45
HSD17B10 Q99714 3/20 0.45
MAPT P10636 3/20 0.45
GLA P06280 2/20 0.45
HPGD P15428 2/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
ATM Q13315 1/20 0.45
CFTR P13569 2/20 0.44
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
SOS1 Q07889 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31546995 0.93 GAA (0.53) GAAABL1NQO2KDM4EALDH1A1
SCHEMBL3340065 0.93 GAA (0.53) GAAABL1NQO2KDM4EALDH1A1
SCHEMBL3529471 0.86 ABL1 (0.56) GAAABL1NQO2KDM4EALDH1A1
SCHEMBL9793695 0.85 GAA (0.59) GAAABL1NQO2KDM4EALDH1A1
SCHEMBL23774898 0.84 GAA (0.54) GAAABL1NQO2KDM4EALDH1A1
SCHEMBL8378560 0.84 GAA (0.49) GAAABL1KDM4EALDH1A1MAPT
SCHEMBL17118715 0.84 MAPT (0.47) GAAABL1NQO2ALDH1A1MAPT
SCHEMBL19328721 0.84 GAA (0.72) GAAABL1NQO2KDM4EALDH1A1
SCHEMBL31487952 0.84 MAPT (0.47) GAAABL1NQO2ALDH1A1MAPT
SCHEMBL7762378 0.84 ABL1 (0.61) GAAABL1NQO2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122094953-A 1, 3-Dihydro-2H-pyrrolo [3,4-c ] quinoline derivatives as cGAS inhibitors for the treatment of inflammatory and/or autoimmune diseases 2026-05-26 CN disclosed
WO-2025040569-A1 1,3-DIHYDRO-2H-PYRROLO[3,4-C]QUINOLINE DERIVATIVES AS CGAS INHIBITORS FOR THE TREATMENT OF INFLAMMATORY AND/OR AUTOIMMUNE DISEASES KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2025-02-27 WO disclosed
US-10189843-B2 Fused pyrazole derivative having autotaxin inhibitory activity THE UNIVERSITY OF TOKYO (JP) 2019-01-29 US disclosed
US-10150787-B2 TC-PTP inhibitors as APC activators for immunotherapy THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIVERSITY (CA) 2018-12-11 US disclosed
US-20180265531-A1 TC-PTP INHIBITORS AS APC ACTIVATORS FOR IMMUNOTHERAPY THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIVERSITY (CA) 2018-09-20 US disclosed
US-10005804-B2 TC-PTP inhibitors as APC activators for immunotherapy THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING / MCGILL UNIV (CA) 2018-06-26 US disclosed
US-10005804-B2 TC-PTP inhibitors as APC activators for immunotherapy THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING / MCGILL UNIV (CA) 2018-06-26 US disclosed
US-20180072763-A1 TC-PTP INHIBITORS AS APC ACTIVATORS FOR IMMUNOTHERAPY THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING / MCGILL UNIV (CA) 2018-03-15 US disclosed
US-20180072763-A1 TC-PTP INHIBITORS AS APC ACTIVATORS FOR IMMUNOTHERAPY THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING / MCGILL UNIV (CA) 2018-03-15 US disclosed
US-9828399-B2 TC-PTP inhibitors as APC activators for immunotherapy THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIVERSITY (CA) 2017-11-28 US disclosed
US-9828399-B2 TC-PTP inhibitors as APC activators for immunotherapy THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING/MCGILL UNIVERSITY (CA) 2017-11-28 US disclosed
US-20170015690-A1 TC-PTP INHIBITORS AS APC ACTIVATORS FOR IMMUNOTHERAPY THE ROYAL INSTITUTE FOR THE ADVANCEMENT OF LEARNING / MCGILL UNIVERSITY (CA) 2017-01-19 US disclosed
US-20170015690-A1 TC-PTP INHIBITORS AS APC ACTIVATORS FOR IMMUNOTHERAPY THE ROYAL INSTITUTE FOR THE ADVANCEMENT OF LEARNING / MCGILL UNIVERSITY (CA) 2017-01-19 US disclosed
US-20170015690-A1 TC-PTP INHIBITORS AS APC ACTIVATORS FOR IMMUNOTHERAPY THE ROYAL INSTITUTE FOR THE ADVANCEMENT OF LEARNING / MCGILL UNIVERSITY (CA) 2017-01-19 US disclosed
EP-3110824-A1 TC-PTP INHIBITORS AS APC ACTIVATORS FOR IMMUNOTHERAPY The Royal Institution for the Advancement of Learning / McGill University (CA) 2017-01-04 EP disclosed
US-20160376278-A1 FUSED PYRAZOLE DERIVATIVE HAVING AUTOTAXIN INHIBITORY ACTIVITY THE UNIVERSITY OF TOKYO (JP) 2016-12-29 US disclosed
WO-2015127548-A1 TC-PTP INHIBITORS AS APC ACTIVATORS FOR IMMUNOTHERAPY THE ROYAL INSTITUTION FOR THE ADVANCEMENT OF LEARNING / MCGILL UNIVERSITY (CA) 2015-09-03 WO disclosed
US-20070196270-A1 Compounds As Ccri Antagonists HENG RICHARD 2007-08-23 US disclosed
US-20070196270-A1 Compounds As Ccri Antagonists HENG RICHARD 2007-08-23 US disclosed
US-20070196270-A1 Compounds As Ccri Antagonists HENG RICHARD 2007-08-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10005804-B2 TC-PTP inhibitors as APC activators for immunotherapy PTPRCAP, PTPRC, PTPA GAA 373/4885ABL1 422/4885NQO2 4277/4885
US-10189843-B2 Fused pyrazole derivative having autotaxin inhibitory activity ENPP2, PRTN3, TPX2 GAA 1152/4885ABL1 4664/4885NQO2 936/4885
US-20170015690-A1 TC-PTP INHIBITORS AS APC ACTIVATORS FOR IMMUNOTHERAPY PTPRCAP, PTPRC, PTPA GAA 373/4885ABL1 422/4885NQO2 4277/4885
US-20180265531-A1 TC-PTP INHIBITORS AS APC ACTIVATORS FOR IMMUNOTHERAPY PTPRCAP, PTPRC, PTPA GAA 373/4885ABL1 422/4885NQO2 4277/4885
US-20160376278-A1 FUSED PYRAZOLE DERIVATIVE HAVING AUTOTAXIN INHIBITORY ACTIVITY ENPP2, PRTN3, TPX2 GAA 1152/4885ABL1 4664/4885NQO2 936/4885
US-20180072763-A1 TC-PTP INHIBITORS AS APC ACTIVATORS FOR IMMUNOTHERAPY PTPRCAP, PTPRC, PTPA GAA 373/4885ABL1 422/4885NQO2 4277/4885
US-10150787-B2 TC-PTP inhibitors as APC activators for immunotherapy PTPRCAP, PTPRC, PTPA GAA 373/4885ABL1 422/4885NQO2 4277/4885
US-20070196270-A1 Compounds As Ccri Antagonists CCR1, CCR10, CCR4 GAA 2746/4885ABL1 2299/4885NQO2 2776/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.