SCHEMBL5597526

SCHEMBL5597526

Nc1c(Br)cc(C[C@@H](NC(=O)N2CCC(N3Cc4ccc(OC(=O)O)cc4NC3=O)CC2)C(=O)[N+]2(C3CCNCC3)CCCCC2)cc1Br

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CALCA P06881 2/20 0.47
CALCRL Q16602 18/20 0.46
CYP3A4 P08684 14/20 0.46
RAMP1 O60894 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6270466 0.75 CALCA (0.61) CALCACALCRLCYP3A4RAMP1
SCHEMBL3876511 0.75 CALCA (0.71) CALCACALCRLCYP3A4RAMP1
SCHEMBL4586249 0.75 CALCRL (0.59) CALCACALCRLCYP3A4RAMP1
SCHEMBL4717830 0.75 CALCRL (0.49) CALCACALCRLCYP3A4RAMP1
SCHEMBL3965813 0.75 CALCRL (0.64) CALCACALCRLCYP3A4RAMP1
SCHEMBL3960011 0.74 CALCRL (0.66) CALCRLCYP3A4
SCHEMBL3959637 0.73 CALCRL (0.67) CALCRLCYP3A4
SCHEMBL4585961 0.73 CALCRL (0.47) CALCACALCRLCYP3A4
SCHEMBL6272723 0.73 CALCA (0.63) CALCACALCRLCYP3A4RAMP1
SCHEMBL6267999 0.73 CALCA (0.63) CALCACALCRLCYP3A4RAMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833478-A1 USE OF SELECTED CGRP ANTAGONISTS IN COMBINATION WITH OTHER ANTIMIGRAINE MEDICAL SUBSTANCES FOR THE TREATMENT OF MIGRAINE Boehringer Ingelheim International GmbH (DE) 2007-09-19 EP claimed
WO-2006072413-A1 USE OF SELECTED CGRP ANTAGONISTS IN COMBINATION WITH OTHER ANTIMIGRAINE MEDICAL SUBSTANCES FOR THE TREATMENT OF MIGRAINE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-07-13 WO claimed