SCHEMBL5598041

SCHEMBL5598041

Cc1ccc(Cn2c(-c3cccc(-c4ccc5ccn(C(=O)OCC(C)C)c5c4)c3)cc(C(F)(F)F)c(C#N)c2=O)c(C)c1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 4/20 0.40
NR1H3 Q13133 4/20 0.40
RXRA P19793 3/20 0.40
TNKS O95271 3/20 0.32
TNKS2 Q9H2K2 3/20 0.32
CYP2C9 P11712 2/20 0.31
CYP2C19 P33261 2/20 0.31
CYP3A4 P08684 1/20 0.31
POLQ O75417 3/20 0.31
RXFP1 Q9HBX9 2/20 0.31
MAPT P10636 2/20 0.31
POLB P06746 1/20 0.31
XDH P47989 1/20 0.30
PDE4D Q08499 1/20 0.30
MCHR1 Q99705 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5598162 0.95 NR1H2 (0.40) NR1H2NR1H3RXRATNKSTNKS2
SCHEMBL5795184 0.90 RXRA (0.45) NR1H2NR1H3RXRAMAPTPOLB
SCHEMBL4899624 0.90 NR1H2 (0.41) NR1H2NR1H3RXRATNKSTNKS2
SCHEMBL4897419 0.84 NR1H2 (0.42) NR1H2NR1H3RXRATNKSTNKS2
SCHEMBL4907759 0.84 NR1H2 (0.43) NR1H2NR1H3RXRATNKSTNKS2
SCHEMBL5598263 0.83 NR1H2 (0.39) NR1H2NR1H3RXRATNKSTNKS2
SCHEMBL4908027 0.80 NR1H2 (0.47) NR1H2NR1H3RXRATNKSTNKS2
SCHEMBL5823324 0.80 NR1H2 (0.43) NR1H2NR1H3RXRATNKSTNKS2
SCHEMBL4897626 0.79 RXRA (0.46) NR1H2NR1H3RXRAMAPTPOLB
SCHEMBL4907807 0.79 NR1H2 (0.47) NR1H2NR1H3RXRATNKSTNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773337-A2 MODULATORS OF NUCLEAR RECEPTORS Exelixis, Inc. (US) 2007-04-18 EP disclosed
WO-2006025979-A9 MODULATORS OF NUCLEAR RECEPTORS EXELIXIS INC (US) 2006-04-20 WO disclosed
WO-2006025979-A2 MODULATORS OF NUCLEAR RECEPTORS EXELIXIS, INC. (US) 2006-03-09 WO disclosed