SCHEMBL5598263

SCHEMBL5598263

Cc1ccc(Cn2c(-c3cccc(-c4cnn(C(=O)OCC(C)C)c4)c3)cc(C(F)(F)F)c(C#N)c2=O)c(C)c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 4/20 0.39
NR1H3 Q13133 4/20 0.39
RXRA P19793 3/20 0.39
POLQ O75417 5/20 0.33
TNKS O95271 2/20 0.33
TNKS2 Q9H2K2 2/20 0.33
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
PPARD Q03181 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4E B2RXH2 2/20 0.31
CSF1R P07333 1/20 0.31
KIT P10721 1/20 0.31
GLA P06280 1/20 0.31
CHRM1 P11229 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4904604 0.89 NR1H2 (0.41) NR1H2NR1H3RXRAPOLQTNKS
SCHEMBL5598162 0.84 NR1H2 (0.40) NR1H2NR1H3RXRAPOLQTNKS
SCHEMBL4902577 0.83 NR1H2 (0.45) NR1H2NR1H3RXRATNKSTNKS2
SCHEMBL5598041 0.83 NR1H2 (0.40) NR1H2NR1H3RXRAPOLQTNKS
SCHEMBL4907972 0.83 NR1H2 (0.41) NR1H2NR1H3RXRATNKSTNKS2
SCHEMBL14184099 0.83 MEN1 (0.42) NR1H2NR1H3RXRAPOLQRXFP1
SCHEMBL4908434 0.82 RXRA (0.42) NR1H2NR1H3RXRATNKSTNKS2
SCHEMBL4902212 0.80 RXRA (0.44) NR1H2NR1H3RXRARXFP1KDM4E
SCHEMBL4901856 0.79 NR1H2 (0.47) NR1H2NR1H3RXRATNKSTNKS2
SCHEMBL4907881 0.79 NR1H2 (0.46) NR1H2NR1H3RXRACYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773337-A2 MODULATORS OF NUCLEAR RECEPTORS Exelixis, Inc. (US) 2007-04-18 EP disclosed
WO-2006025979-A9 MODULATORS OF NUCLEAR RECEPTORS EXELIXIS INC (US) 2006-04-20 WO disclosed
WO-2006025979-A2 MODULATORS OF NUCLEAR RECEPTORS EXELIXIS, INC. (US) 2006-03-09 WO disclosed