SCHEMBL5598902

SCHEMBL5598902

CC(Cn1ccnc1C(COCCCN(C)C)c1ccc(Cl)cc1)N1CCCCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 11/20 0.39
HRH3 Q9Y5N1 10/20 0.39
SLC6A2 P23975 7/20 0.34
SLC6A3 Q01959 6/20 0.34
CHRM2 P08172 3/20 0.34
ADRA2B P18089 3/20 0.34
HRH1 P35367 3/20 0.34
KCNH2 Q12809 3/20 0.34
CHRM5 P08912 2/20 0.34
CHRM1 P11229 2/20 0.34
HRH2 P25021 2/20 0.34
HTR2A P28223 2/20 0.34
CYP2D6 P10635 2/20 0.34
SIGMAR1 Q99720 2/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
NFKB1 P19838 1/20 0.34
THPO P40225 1/20 0.34
ADRA1A P35348 1/20 0.34
SCN1A P35498 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6650426 0.76 HRH3 (0.33) SLC6A4HRH3SLC6A2SLC6A3
SCHEMBL4905451 0.75 HRH3 (0.39) SLC6A4HRH3SLC6A2SLC6A3CHRM2
SCHEMBL5599833 0.74 HRH3 (0.39) SLC6A4HRH3SLC6A2SLC6A3
SCHEMBL5924545 0.72 HRH3 (0.43) SLC6A4HRH3SLC6A2SLC6A3CHRM2
SCHEMBL4910298 0.71 HRH3 (0.40) SLC6A4HRH3SLC6A2SLC6A3CHRM2
SCHEMBL5602140 0.70 HRH3 (0.36) SLC6A4HRH3SLC6A2SLC6A3CHRM2
SCHEMBL6648867 0.70 SLC6A4 (0.32) SLC6A4HRH3SLC6A2SLC6A3CYP2D6
SCHEMBL5599393 0.68 PSMB1 (0.40) SLC6A4HRH3SLC6A2SIGMAR1LMNA
SCHEMBL5601418 0.66 FFAR1 (0.44) SLC6A4HRH3L3MBTL1
SCHEMBL4910626 0.64 HRH3 (0.51) SLC6A4HRH3SLC6A2SLC6A3CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1755678-A2 ACTIVE SUBSTANCE COMBINATION OF A CARBINOL COMPOUND AND AN OPIOID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-02-28 EP disclosed
WO-2005097192-A2 ACTIVE SUBSTANCE COMBINATION OF A CARBINOL COMPOUND AND AN OPIOID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2005-10-20 WO disclosed