SCHEMBL5599146

SCHEMBL5599146

Cn1ccnc1Cc1cccc(C(O)Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 2/20 0.46
KDM4E B2RXH2 1/20 0.41
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
MAPT P10636 1/20 0.38
CBLB Q13191 5/20 0.35
POLB P06746 1/20 0.34
FDPS P14324 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6650689 0.83 L3MBTL1 (0.40) OPRK1KDM4EKMT2AMEN1MAPT
SCHEMBL6650490 0.80 MEN1 (0.37) OPRK1KDM4EKMT2AMEN1MAPT
SCHEMBL6649435 0.78 OPRK1 (0.37) OPRK1KDM4EKMT2AMEN1POLB
SCHEMBL20204951 0.77 CYP11B1 (0.45) OPRK1KMT2AMEN1MAPTPOLB
SCHEMBL6651103 0.76 OPRK1 (0.36) OPRK1KDM4EKMT2AMEN1MAPT
SCHEMBL25183645 0.76 CYP11B1 (0.44) OPRK1KMT2AMEN1MAPTPOLB
SCHEMBL30374060 0.76 CYP11B1 (0.44) OPRK1KMT2AMEN1MAPTPOLB
SCHEMBL1044189 0.74 KMT2A (0.54) KDM4EKMT2AMEN1MAPTFDPS
SCHEMBL6651257 0.73 KMT2A (0.44) OPRK1KDM4EKMT2AMEN1MAPT
Hydrochloric Acid SCHEMBL1875423 0.73 KMT2A (0.53) KDM4EKMT2AMEN1MAPTFDPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1103243-B1 UTILIZATION OF ARYL(OR HETEROARYL)AZOLYLCARBINOL DERIVATIVES FOR THE TREATMENT OF TROUBLES MEDIATED BY AN EXCESS OF SUBSTANCE P ESTEVE LABOR DR (ES) 2004-01-07 EP claimed
EP-1755678-A2 ACTIVE SUBSTANCE COMBINATION OF A CARBINOL COMPOUND AND AN OPIOID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-02-28 EP disclosed
WO-2005097192-A2 ACTIVE SUBSTANCE COMBINATION OF A CARBINOL COMPOUND AND AN OPIOID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2005-10-20 WO disclosed