SCHEMBL5599295

SCHEMBL5599295

C=CC[C@H]1N(C(=O)c2ccc3c(c2)OCO3)c2ccc(F)cc2C12CCNCC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
NR3C2 P08235 9/20 0.38
CTNNB1 P35222 1/20 0.37
WNT3A P56704 1/20 0.37
SHMT2 P34897 1/20 0.36
NR3C1 P04150 5/20 0.36
PGR P06401 3/20 0.36
ALDH1A1 P00352 3/20 0.36
MAPT P10636 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 2/20 0.36
GAA P10253 1/20 0.36
CASP3 P42574 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5783881 0.87 TSHR (0.49) TSHRL3MBTL1NR3C2CTNNB1WNT3A
SCHEMBL5599105 0.83 CHRNB2 (0.34) NR3C2NR3C1
SCHEMBL5780824 0.83 GNRHR (0.37)
SCHEMBL5599115 0.83 GNRHR (0.34) NR3C2NR3C1
SCHEMBL5788788 0.82 ALDH1A1 (0.38) TSHRL3MBTL1ALDH1A1MAPTGAA
SCHEMBL5599768 0.81 GNRHR (0.36)
SCHEMBL5780470 0.81 MAPK1 (0.37) MAPT
SCHEMBL5599622 0.81 MAPK1 (0.37) MAPT
SCHEMBL5786885 0.81 GNRHR (0.33) KDM4E
SCHEMBL5783676 0.81 ALDH1A1 (0.46) TSHRALDH1A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO claimed