SCHEMBL5599115

SCHEMBL5599115

C=CC[C@H]1N(C(=O)c2ccc(F)c(C(F)(F)F)c2)c2ccc(F)cc2C12CCNCC2

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GNRHR P30968 2/20 0.34
HSD11B1 P28845 1/20 0.33
KCNH2 Q12809 1/20 0.32
PSEN1 P49768 6/20 0.32
PSEN2 P49810 6/20 0.32
APH1B Q8WW43 6/20 0.32
NCSTN Q92542 6/20 0.32
APH1A Q96BI3 6/20 0.32
PSENEN Q9NZ42 6/20 0.32
TAS1R3 Q7RTX0 2/20 0.32
TAS1R1 Q7RTX1 2/20 0.32
TAS1R2 Q8TE23 2/20 0.32
NR3C2 P08235 2/20 0.32
VNN1 O95497 1/20 0.31
PDE4B Q07343 1/20 0.31
SLC6A2 P23975 2/20 0.30
SLC6A4 P31645 2/20 0.30
NR3C1 P04150 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5781400 0.87 HSD11B1 (0.35) GNRHRHSD11B1KCNH2PSEN1PSEN2
SCHEMBL5780824 0.85 GNRHR (0.37) GNRHRKCNH2PSEN1PSEN2APH1B
SCHEMBL5599295 0.83 TSHR (0.47) NR3C2NR3C1
SCHEMBL5786885 0.83 GNRHR (0.33) GNRHRKCNH2PSEN1PSEN2APH1B
SCHEMBL5788788 0.82 ALDH1A1 (0.38) GNRHRHSD11B1KCNH2
SCHEMBL5599768 0.81 GNRHR (0.36) GNRHRKCNH2PSEN1PSEN2APH1B
SCHEMBL5599105 0.81 CHRNB2 (0.34) GNRHRKCNH2NR3C2NR3C1
SCHEMBL5599622 0.81 MAPK1 (0.37) GNRHRKCNH2PSEN1PSEN2APH1B
SCHEMBL5780470 0.81 MAPK1 (0.37) GNRHRKCNH2PSEN1PSEN2APH1B
SCHEMBL5783676 0.81 ALDH1A1 (0.46) GNRHRHSD11B1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO claimed