SCHEMBL5599306

SCHEMBL5599306

CC(C)(C)OC(=O)[C@H]1c2ccccc2C2(CCNCC2)CN1C(=O)C(c1ccccc1)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
AGTR2 P50052 5/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
NR1H2 P55055 3/20 0.32
RXRA P19793 2/20 0.32
NR1H3 Q13133 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5599646 0.76 AGTR2 (0.34) USP2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL13689881 0.72 KDM1A (0.37) CYP3A4CYP2C9
SCHEMBL4116754 0.72 ACE (0.35) USP2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4116886 0.72 HSD11B1 (0.41) HDAC1HDAC8HDAC6NR1H2RXRA
Hydrochloric Acid SCHEMBL1747690 0.71 NOTUM (0.34) USP2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL3994423 0.69 DPP9 (0.35) USP2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5599645 0.69 NOTUM (0.51) USP2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4124959 0.69 HSD11B1 (0.39)
SCHEMBL5578840 0.67 DPP9 (0.44) USP2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5578573 0.66 HDAC1 (0.50) HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO claimed