SCHEMBL5599378

SCHEMBL5599378

CC(=C(C#N)C#N)c1ccc(O)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.54
ESR2 Q92731 5/20 0.54
CYP19A1 P11511 2/20 0.45
CA12 O43570 1/20 0.41
CA2 P00918 1/20 0.41
CA3 P07451 1/20 0.41
CA6 P23280 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
HSD17B1 P14061 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRB2 P47870 1/20 0.40
NQO2 P16083 1/20 0.40
MAPT P10636 2/20 0.40
APP P05067 1/20 0.40
SNCA P37840 1/20 0.40
EGFR P00533 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18972851 0.87 ESR1 (0.65) ESR1ESR2CYP19A1
SCHEMBL15626973 0.82 ALDH1A1 (0.41) GABRA1GABRB1GABRG2GABRB3GABRB2
SCHEMBL26859454 0.80 RECQL (0.42) CA2GABRA1GABRB1GABRG2GABRB3
SCHEMBL10154445 0.80 CYP19A1 (0.56) ESR1ESR2CYP19A1CA3CA6
SCHEMBL28354801 0.80 APP (0.42) CA2GABRA1GABRB1GABRG2GABRB3
SCHEMBL4657618 0.80 GABRA1 (0.56) CA2GABRA1GABRB1GABRG2GABRB3
SCHEMBL178769 0.79 ALDH1A1 (0.48) ESR1GABRA1GABRB1GABRG2GABRB3
Dimethylstilbestrol SCHEMBL125635 0.77 ESR1 (0.74) ESR1ESR2CYP19A1CA12CA2
Dimethylstilbestrol SCHEMBL13339102 0.77 ESR1 (0.74) ESR1ESR2CYP19A1CA12CA2
Dimethylstilbestrol SCHEMBL125634 0.77 ESR1 (0.74) ESR1ESR2CYP19A1CA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1764363-A2 SUBSTITUTED ACETOPHENONEDERIVATIVES Riemser Arzneimittel AG (DE) 2007-03-21 EP claimed
EP-1764363-A2 SUBSTITUTED ACETOPHENONEDERIVATIVES Riemser Arzneimittel AG (DE) 2007-03-21 EP disclosed
US-4783280-A Liquid crystal mixture HOFFMANN-LA ROCHE INC. (US) 1988-11-08 US disclosed
US-4460770-A Liquid crystal mixture HOFFMANN-LA ROCHE INC. (US) 1984-07-17 US disclosed