SCHEMBL5599576

SCHEMBL5599576

CC(c1ccc(OCC(Cl)N(C)C)cc1)c1nccn1CCN1CCCCC1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PSMB1 P20618 1/20 0.48
PSMB5 P28074 1/20 0.48
KMT2A Q03164 4/20 0.40
MEN1 O00255 2/20 0.40
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
TSHR P16473 1/20 0.38
HRH3 Q9Y5N1 11/20 0.37
SLC6A4 P31645 9/20 0.37
LTA4H P09960 1/20 0.37
SLC6A2 P23975 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5600674 0.91 PSMB1 (0.51) PSMB1PSMB5KMT2AMEN1ALDH1A1
SCHEMBL5599393 0.77 PSMB1 (0.40) PSMB1PSMB5KMT2AMEN1ALDH1A1
SCHEMBL5600030 0.66 CYP3A4 (0.43) KMT2AMEN1TSHRHRH3SLC6A4
SCHEMBL6655024 0.65 PSMB1 (0.78) PSMB1PSMB5KMT2AMEN1ALDH1A1
SCHEMBL5601407 0.64 MEN1 (0.44) KMT2AMEN1LMNAMAPTTSHR
SCHEMBL5599453 0.64 HRH3 (0.43) PSMB1PSMB5HRH3SLC6A4LTA4H
SCHEMBL5599192 0.64 LMNA (0.36) KMT2ALMNAMAPT
SCHEMBL12204133 0.63 PSMB1 (0.83) PSMB1PSMB5KMT2AMEN1ALDH1A1
SCHEMBL8697896 0.62 KMT2A (0.53) KMT2AALDH1A1TSHRHRH3
SCHEMBL6654256 0.62 MEN1 (0.33) KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1755678-A2 ACTIVE SUBSTANCE COMBINATION OF A CARBINOL COMPOUND AND AN OPIOID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-02-28 EP disclosed
WO-2005097192-A2 ACTIVE SUBSTANCE COMBINATION OF A CARBINOL COMPOUND AND AN OPIOID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2005-10-20 WO disclosed