SCHEMBL5599671

SCHEMBL5599671

C=CC[C@@H]1c2ccccc2C2(CCNCC2)CN1C(=O)c1c(F)cccc1F

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
HTR6 P50406 1/20 0.32
LMNA P02545 2/20 0.31
GAA P10253 1/20 0.31
PREP P48147 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
P2RY1 P47900 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5599341 0.90 TSHR (0.33) KMT2AMEN1HTR6LMNAGAA
SCHEMBL5599440 0.85 MCHR2 (0.33) KMT2AMEN1
SCHEMBL5599346 0.83 KMT2A (0.37) KMT2ACHRM3GAA
SCHEMBL5599778 0.77 KMT2A (0.39) KMT2AMEN1LMNA
SCHEMBL5599143 0.76 CYP2C9 (0.37) CYP1A2CYP2C9CYP2C19
SCHEMBL5599653 0.75 KMT2A (0.41) KMT2AMEN1LMNAGAAMAPT
SCHEMBL5781243 0.72 CYP1A2 (0.36) KMT2ACHRM1CHRM3LMNACYP1A2
SCHEMBL5578434 0.66 HDAC1 (0.46) CYP1A2CYP2C9CYP2C19
SCHEMBL4116754 0.66 ACE (0.35) CYP1A2CYP2C9P2RY1
SCHEMBL3994423 0.65 DPP9 (0.35) KMT2ACYP1A2CYP2C9P2RY1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO claimed