SCHEMBL5599734

SCHEMBL5599734

CCc1cccc(C(N)=O)c1C1CCOCC1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
TYK2 P29597 1/20 0.40
JAK3 P52333 1/20 0.40
HTR1A P08908 3/20 0.39
PARP1 P09874 8/20 0.38
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5599187 0.85 HTR1A (0.41) HTR1APARP1KDM4E
Hydrochloric Acid SCHEMBL27801407 0.84 HTR1A (0.40) HTR1APARP1KDM4E
SCHEMBL20822489 0.82 CYP11B1 (0.42) CYP11B1CYP11B2JAK2JAK1TYK2
SCHEMBL5599730 0.79 PARP1 (0.40) CYP11B1CYP11B2JAK2JAK1TYK2
SCHEMBL17185049 0.74 PARP1 (0.46) CYP11B1CYP11B2PARP1
SCHEMBL2976919 0.74 KDM4E (0.45) HTR1APARP1KDM4EALDH1A1
SCHEMBL28470220 0.74 MAPK1 (0.39) CYP11B1CYP11B2JAK2JAK1TYK2
SCHEMBL20822490 0.74 PARP1 (0.43) CYP11B1CYP11B2PARP1
SCHEMBL16956335 0.73 GABRA1 (0.41)
SCHEMBL27811001 0.73 BID (0.40) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740584-A1 FUSED QUINOLINE DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-01-10 EP disclosed
WO-2005105802-A1 FUSED QUINOLINE DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-11-10 WO disclosed