SCHEMBL5599800

SCHEMBL5599800

O=C(O)Nc1nc(CC(=O)Nc2ccccc2O)cs1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.58
KDM4E B2RXH2 2/20 0.58
GAA P10253 1/20 0.58
MEN1 O00255 4/20 0.57
KMT2A Q03164 4/20 0.57
MAPT P10636 4/20 0.55
ALDH1A1 P00352 3/20 0.55
ALOX12 P18054 3/20 0.55
LMNA P02545 2/20 0.55
PDE5A O76074 6/20 0.55
SLC12A2 P55011 1/20 0.54
SLC12A5 Q9H2X9 1/20 0.54
CYP1A2 P05177 2/20 0.54
CYP3A4 P08684 2/20 0.54
CYP2D6 P10635 2/20 0.54
CYP2C9 P11712 2/20 0.54
CYP2C19 P33261 2/20 0.54
ITGB1 P05556 1/20 0.51
ITGA4 P13612 1/20 0.51
PDE1A P54750 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3597144 0.86 SMN1; SMN2 (0.57) SMN1; SMN2KDM4EGAAMEN1KMT2A
SCHEMBL3607475 0.78 PDE5A (0.70) KDM4EPDE5APDE1APDE1BPDE1C
SCHEMBL5604178 0.78 MEN1 (0.61) KDM4EGAAMEN1KMT2AMAPT
SCHEMBL8249057 0.77 HDAC1 (0.53) SMN1; SMN2KDM4EGAAMEN1KMT2A
SCHEMBL5599931 0.75 PDE5A (0.53) SMN1; SMN2KDM4EGAAMEN1KMT2A
SCHEMBL17444763 0.73 MEN1 (0.81) SMN1; SMN2KDM4EGAAMEN1KMT2A
SCHEMBL25720785 0.73 PDE5A (0.79) SMN1; SMN2KDM4EMEN1KMT2AMAPT
SCHEMBL92487 0.72 ELOVL1 (0.65) GAAMEN1KMT2ALMNAPDE5A
SCHEMBL5155280 0.71 ITGB1 (0.77) SMN1; SMN2GAAMAPTALDH1A1LMNA
SCHEMBL465934 0.71 SMN1; SMN2 (0.51) SMN1; SMN2KDM4EGAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007017728-A2 NOVEL HETEROCYCLIC COMPOUNDS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-02-15 WO claimed
WO-2007017728-A2 NOVEL HETEROCYCLIC COMPOUNDS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-02-15 WO disclosed