SCHEMBL5604178

SCHEMBL5604178

O=C(O)Nc1nc(CC(=O)Nc2cccc(O)c2)cs1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.61
KMT2A Q03164 1/20 0.61
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
CTPS1 P17812 9/20 0.55
GAA P10253 1/20 0.52
MAPT P10636 1/20 0.52
NLRP3 Q96P20 1/20 0.51
PDE5A O76074 2/20 0.50
KDM4E B2RXH2 1/20 0.50
PDE1A P54750 1/20 0.50
PDE1B Q01064 1/20 0.50
PDE1C Q14123 1/20 0.50
EGFR P00533 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8249060 0.79 MEN1 (0.49) MEN1KMT2ACTPS1MAPTPDE5A
SCHEMBL5599800 0.78 SMN1; SMN2 (0.58) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL25720785 0.76 PDE5A (0.79) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL3607475 0.76 PDE5A (0.70) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL3597144 0.74 SMN1; SMN2 (0.57) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL11516149 0.74 PDE5A (0.64) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL5599931 0.73 PDE5A (0.53) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL10977240 0.72 MAPT (0.71) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL3599789 0.72 MAPT (0.46) GAAMAPTNLRP3EGFR
SCHEMBL11517104 0.72 PDE5A (0.62) MEN1KMT2ACYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007017728-A2 NOVEL HETEROCYCLIC COMPOUNDS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-02-15 WO claimed
WO-2007017728-A2 NOVEL HETEROCYCLIC COMPOUNDS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-02-15 WO disclosed