SCHEMBL5606609

SCHEMBL5606609

O=P(O)(O)OC1=CCCc2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 2/20 0.43
SRC P12931 3/20 0.40
CES1 P23141 1/20 0.37
L3MBTL1 Q9Y468 3/20 0.35
HPGD P15428 2/20 0.35
ACP3 P15309 1/20 0.35
MAPT P10636 3/20 0.35
INPPL1 O15357 1/20 0.34
INPP5B P32019 1/20 0.34
INPP5A Q14642 1/20 0.34
CYP2A6 P11509 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
USP2 O75604 1/20 0.34
PDE3A Q14432 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5606605 0.86 GPR84 (0.45) GPR84CES1L3MBTL1HPGDMAPT
SCHEMBL5606866 0.80 GPR84 (0.40) GPR84SRCCES1L3MBTL1HPGD
SCHEMBL8500693 0.77 MAPT (0.44) CES1L3MBTL1HPGDMAPTALDH1A1
SCHEMBL5607172 0.76 MPO (0.54) L3MBTL1MAPTALDH1A1KDM4ENPC1
SCHEMBL27532472 0.74 MAPT (0.46) L3MBTL1HPGDMAPTALDH1A1HSD17B10
SCHEMBL10782148 0.74 CES1 (0.41) GPR84CES1L3MBTL1HPGDACP3
SCHEMBL19096363 0.74 CES1 (0.41) GPR84CES1L3MBTL1HPGDMAPT
SCHEMBL13160775 0.73 MAPT (0.35) CES1L3MBTL1MAPTALDH1A1KMT2A
SCHEMBL6161470 0.73 CES1 (0.39) CES1L3MBTL1HPGDMAPTCYP2A6
SCHEMBL27677730 0.72 CES1 (0.39) GPR84CES1L3MBTL1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2005528450-A 2005-09-22 JP claimed
EP-1509484-A2 PROCESS FOR PREPARING VINYLAROMATIC COMPOUNDS DSM IP Assets B.V. (NL) 2005-03-02 EP claimed
WO-2003102202-A2 PROCESS FOR PREPARING VINYLAROMATIC COMPOUNDS DSM IP ASSETS B.V. (NL) 2003-12-11 WO claimed
US-6608212-B1 Palladium catalyzed coupling of a vinylphosphate and aryl-metal halide; preparation of such as 1-(4-(2-(pyrrolidin-n-yl)-ethoxy)phenyl)-6-methoxy-3,4-dihydronaphthalene PFIZER, INC. 2003-08-19 US claimed
EP-1754709-A1 Process for preparing vinylphosphates DSM IP Assets B.V. (NL) 2007-02-21 EP disclosed
EP-1509484-A2 PROCESS FOR PREPARING VINYLAROMATIC COMPOUNDS DSM IP Assets B.V. (NL) 2005-03-02 EP disclosed
WO-2003102202-A2 PROCESS FOR PREPARING VINYLAROMATIC COMPOUNDS DSM IP ASSETS B.V. (NL) 2003-12-11 WO disclosed
US-6608212-B1 Palladium catalyzed coupling of a vinylphosphate and aryl-metal halide; preparation of such as 1-(4-(2-(pyrrolidin-n-yl)-ethoxy)phenyl)-6-methoxy-3,4-dihydronaphthalene PFIZER, INC. 2003-08-19 US disclosed