SCHEMBL56080

SCHEMBL56080

OC1CCC2(CCCO2)CC1

nearest known ligand 0.36

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.36
GPR119 Q8TDV5 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17304275 1.00 TSHR (0.36) TSHRGPR119
SCHEMBL5307808 0.95 GPR119 (0.34) TSHRGPR119
SCHEMBL31032139 0.90 TSHR (0.33) TSHR
SCHEMBL8181997 0.86 OPRK1 (0.33)
SCHEMBL26444547 0.78
SCHEMBL126707 0.78
SCHEMBL126686 0.78
SCHEMBL127016 0.78
SCHEMBL6550937 0.76
SCHEMBL320777 0.75 KCNH2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 118 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025106910-A1 DEGRADER MOLECULES TARGETING ANDROGEN RECEPTOR FLARE THERAPEUTICS INC. (US) 2025-05-22 WO disclosed
EP-4355748-A1 SUBSTITUTED PYRROLO[2,3-D]PYRIMIDINES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION SANOFI (FR) 2024-04-24 EP disclosed
EP-4352055-A1 O-LINKED THIADIAZOLYL COMPOUNDS AS DNA POLYMERASE THETA INHIBITORS Ideaya Biosciences, Inc. (US) 2024-04-17 EP disclosed
WO-2023165570-A1 CYCLOALKYL OR HETEROCYCLYL SUBSTITUTED HETEROARYL COMPOUND, AND COMPOSITION AND USE THEREOF 深圳市塔吉瑞生物医药有限公司 2023-09-07 WO disclosed
WO-2022263472-A1 SUBSTITUTED PYRROLO[2,3-D]PYRIMIDINES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION SANOFI (FR) 2022-12-22 WO disclosed
WO-2022259204-A1 O-LINKED THIADIAZOLYL COMPOUNDS AS DNA POLYMERASE THETA INHIBITORS IDEAYA BIOSCIENCES, INC. (US) 2022-12-15 WO disclosed
EP-3807251-A1 PHENYL AND PYRIDINYL SUBSTITUTED IMIDAZOLES AS MODULATORS OF RORYT Janssen Pharmaceutica NV (BE) 2021-04-21 EP disclosed
EP-3652179-A1 INHIBITORS OF LEUCINE RICH REPEAT KINASE 2 GlaxoSmithKline Intellectual Property Development Ltd (GB) 2020-05-20 EP disclosed
EP-3642195-A1 SUBSTITUTED 5-CYANOINDOLE COMPOUNDS AND USES THEREOF Novartis AG (CH) 2020-04-29 EP disclosed
WO-2019244000-A1 PHENYL AND PYRIDINYL SUBSTITUTED IMIDAZOLES AS MODULATORS OF RORYT JANSSEN PHARMACEUTICA NV (BE) 2019-12-26 WO disclosed
EP-1487778-A1 SUBSTITUTED 4-AMINOCYCLOHEXANOLS Grünenthal GmbH (DE) 2004-12-22 EP disclosed
WO-2003080557-A1 SUBSTITUTED 4-AMINOCYCLOHEXANOLS Grünenthal GmbH (DE) 2003-10-02 WO disclosed
WO-2001072751-A1 PYRROLOPYRIMIDINES AS TYROSINE KINASE INHIBITORS KNOLL GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2001-10-04 WO disclosed
EP-0983225-A1 NEW POLYMERISABLE LIQUID CRYSTALLINE COMPOUNDS Rolic AG (CH) 2000-03-08 EP disclosed
WO-1998052905-A1 NEW POLYMERISABLE LIQUID CRYSTALLINE COMPOUNDS ROLIC AG (CH) 1998-11-26 WO disclosed
EP-0207773-B1 7-[(Substituted)amino]-8-[(substituted)carbonyl)-methylamino]-1-oxaspiro[4.5]decanes as analgesic agents WARNER-LAMBERT COMPANY (US) 1990-01-03 EP disclosed
US-4737493-A 7-((substituted)amino)-8-((substituted)carbonyl)-methylamino)-1-oxaspiro(4,5)decanes as analgesic agents WARNER-LAMBERT COMPANY (US) 1988-04-12 US disclosed
EP-0207773-A2 7-[(Substituted)amino]-8-[(substituted)carbonyl)-methylamino]-1-oxaspiro[4.5]decanes as analgesic agents WARNER-LAMBERT COMPANY (US) 1987-01-07 EP disclosed
US-4508911-A Amine intermediates for analgesic compounds THE UPJOHN COMPANY (US) 1985-04-02 US disclosed
US-4438130-A Analgesic 1-oxa-, aza- and thia-spirocyclic compounds THE UPJOHN COMPANY (US) 1984-03-20 US disclosed