SCHEMBL5608129

SCHEMBL5608129

COc1ccc(N(c2cccc(OC)c2)c2ccccc2OC)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.44
HSD17B1 P14061 1/20 0.42
HSD17B2 P37059 1/20 0.42
MTNR1A P48039 4/20 0.41
MTNR1B P49286 4/20 0.41
NFE2L2 Q16236 1/20 0.40
ENPP2 Q13822 1/20 0.40
CYP1A1 P04798 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP1B1 Q16678 2/20 0.40
ALOX15 P16050 1/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18392045 0.94 MTNR1A (0.43) PTGESHSD17B1HSD17B2MTNR1AMTNR1B
SCHEMBL8943802 0.89 PTGES (0.51) PTGESCYP1A1CYP1A2CYP1B1NPC1
SCHEMBL9163037 0.86 SLC16A3 (0.43) HSD17B1HSD17B2MTNR1AMTNR1BNFE2L2
SCHEMBL8943935 0.85 PTGES (0.51) PTGESCYP1A1CYP1A2CYP1B1ALDH1A1
SCHEMBL23350491 0.85 ALDH1A1 (0.41) HSD17B1HSD17B2MTNR1AMTNR1BMEN1
SCHEMBL28209766 0.84 MTNR1A (0.49) HSD17B1HSD17B2MTNR1AMTNR1BENPP2
SCHEMBL13385303 0.84 CA4 (0.52) HSD17B1HSD17B2MTNR1AMTNR1BENPP2
SCHEMBL8944101 0.84 HSD17B2 (0.50) HSD17B1HSD17B2MTNR1AMTNR1BENPP2
SCHEMBL8944319 0.83 CA12 (0.46) NFE2L2CYP1A1CYP1A2CYP1B1MEN1
SCHEMBL19275049 0.82 CA1 (0.48) PTGESENPP2CYP1A2MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1354887-B1 Ligands for metals and improved metal-catalyzed processes based thereon MASSACHUSETTS INST TECHNOLOGY (US) 2007-04-25 EP disclosed
EP-1354887-B1 Ligands for metals and improved metal-catalyzed processes based thereon MASSACHUSETTS INST TECHNOLOGY (US) 2007-04-25 EP disclosed
EP-1097158-B1 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INST TECHNOLOGY (US) 2006-01-25 EP disclosed