SCHEMBL5608971

SCHEMBL5608971

O=c1c2cc(NS(=O)(=O)c3ccc(F)c(Cl)c3)ccc2[nH]n1CC1CC1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
TSHR P16473 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HTR6 P50406 6/20 0.42
PABPC1 P11940 1/20 0.41
MAPT P10636 2/20 0.41
THRB P10828 1/20 0.41
HTT P42858 1/20 0.41
DRD2 P14416 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
DRD3 P35462 1/20 0.40
BRD4 O60885 2/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1801399 0.87 TP53 (0.44) LMNAHTR6MAPTTHRB
SCHEMBL5608726 0.86 BRD4 (0.53) PKMKMT2AALDH1A1LMNAHTR6
SCHEMBL3915082 0.85 PTGDR2 (0.47) PKMPTGDR2MEN1KMT2AALDH1A1
SCHEMBL1804773 0.83 MEN1 (0.46) PKMPTGDR2MEN1KMT2AALDH1A1
SCHEMBL5617634 0.82 MEN1 (0.49) PKMPTGDR2MEN1KMT2AALDH1A1
SCHEMBL5608793 0.79 PKM (0.41) PKMMEN1KMT2AALDH1A1LMNA
SCHEMBL5608331 0.78 GSPT1 (0.48) PKMMEN1KMT2AALDH1A1LMNA
SCHEMBL1819904 0.73 BRD4 (0.52) PKMLMNAHTR6MAPTHTR2A
SCHEMBL1820048 0.73 ERAP1 (0.46) PKMLMNAMAPTTHRBHTT
SCHEMBL3908576 0.72 PTPN2 (0.42) PKMPTGDR2LMNAMAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797042-A1 INDOZOLONE DERIVATIVES AS 11B-HSD1 INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-06-20 EP disclosed
WO-2006034804-A1 INDOZOLONE DERIVATIVES AS 11B-HSD1 INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2006-04-06 WO disclosed