SCHEMBL5612440

SCHEMBL5612440

Cc1ccccc1-c1nc2nn(-c3ccccc3)cc2c(=O)n1-c1cccc(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.45
THRB P10828 1/20 0.44
TP53 P04637 1/20 0.44
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.41
KCNH2 Q12809 1/20 0.41
GHSR Q92847 1/20 0.41
ADORA3 P0DMS8 2/20 0.39
GAA P10253 1/20 0.39
ADORA2A P29274 1/20 0.38
GRM1 Q13255 1/20 0.38
MAT2A P31153 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5611456 0.85 THRB (0.61) POLBTHRBTP53CYP1A2CYP2D6
SCHEMBL5611548 0.85 TP53 (0.61) POLBTHRBTP53CYP1A2CYP2D6
SCHEMBL5611981 0.83 ADORA3 (0.41) POLBTP53KDM4EALDH1A1LMNA
SCHEMBL1688907 0.83 GRM1 (0.44) KDM4EKMT2AADORA3GRM1
SCHEMBL1689073 0.82 TP53 (0.51) POLBTHRBTP53CYP1A2CYP2D6
SCHEMBL1688973 0.80 KDM4E (0.46) CYP1A2CYP2D6CYP2C9CYP2C19KDM4E
SCHEMBL5611629 0.78 SMN1; SMN2 (0.41) TP53CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL5612509 0.77 MAPT (0.62) POLBTHRBTP53SMN1; SMN2KDM4E
SCHEMBL5611689 0.77 KDM4E (0.43) POLBTP53KDM4EALDH1A1LMNA
SCHEMBL1688982 0.77 KDM4E (0.43) KDM4EADORA3GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807429-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM, LLC (BM) 2007-07-18 EP disclosed
WO-2006047516-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2006-05-04 WO disclosed