Emiglitate

Emiglitate

SCHEMBL5616336

CCOC(=O)c1ccc(OCCN2C[C@H](O)C(O)C(O)[C@H]2CO)cc1

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.48
HRH3 Q9Y5N1 1/20 0.48
GAA P10253 4/20 0.48
GBA2 Q9HCG7 11/20 0.48
GBA1 P04062 4/20 0.48
UGCG Q16739 3/20 0.46
MGAM O43451 2/20 0.46
SI P14410 2/20 0.46
AGL P35573 2/20 0.46
TBXAS1 P24557 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
MAPK1 P28482 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Emiglitate SCHEMBL5188302 1.00 KCNH2 (0.48) KCNH2HRH3GAAGBA2GBA1
Emiglitate SCHEMBL5188305 1.00 KCNH2 (0.48) KCNH2HRH3GAAGBA2GBA1
Emiglitate SCHEMBL26909 1.00 KCNH2 (0.48) KCNH2HRH3GAAGBA2GBA1
SCHEMBL23996617 0.74 GBA2 (0.60) GAAGBA2GBA1UGCGMGAM
SCHEMBL22048754 0.74 KCNH2 (0.57) KCNH2HRH3GAATBXAS1TDP1
SCHEMBL6701399 0.73 TDP1 (0.74) KCNH2HRH3TBXAS1TDP1L3MBTL1
SCHEMBL21408538 0.72 HRH3 (0.79) KCNH2HRH3L3MBTL1MEN1LMNA
SCHEMBL6867384 0.72 TDP1 (0.64) KCNH2HRH3GAATBXAS1TDP1
SCHEMBL9199244 0.72 KCNH2 (0.63) KCNH2HRH3GAATBXAS1TDP1
SCHEMBL6999600 0.71 MAPK1 (0.67) KCNH2HRH3GAATBXAS1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007107843-A1 METHODS OF TREATMENT WITH CETP INHIBITORS PFIZER PRODUCTS INC. (US) 2007-09-27 WO disclosed
WO-2006033001-A1 QUINOLINE COMPOUNDS PFIZER PRODUCTS INC. (US) 2006-03-30 WO disclosed