SCHEMBL9199244

SCHEMBL9199244

CCOC(=O)c1ccc(OCCN2CCNCC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.63
HRH3 Q9Y5N1 1/20 0.63
HRH2 P25021 3/20 0.59
HRH1 P35367 3/20 0.59
KDM4E B2RXH2 3/20 0.55
ALDH1A1 P00352 2/20 0.55
MAPT P10636 2/20 0.55
TDP1 Q9NUW8 2/20 0.55
PSMB1 P20618 1/20 0.52
PSMB5 P28074 1/20 0.52
PSMB2 P49721 1/20 0.52
LTA4H P09960 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
GAA P10253 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.51
TBXAS1 P24557 1/20 0.51
KMT2A Q03164 1/20 0.51
ESR1 P03372 1/20 0.51
ESR2 Q92731 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9200735 0.94 HRH3 (0.72) KCNH2HRH3HRH2HRH1ALDH1A1
SCHEMBL21408538 0.88 HRH3 (0.79) KCNH2HRH3HRH2HRH1KDM4E
SCHEMBL228881 0.87 KCNH2 (0.81) KCNH2HRH3HRH2HRH1KDM4E
SCHEMBL223800 0.87 KCNH2 (0.81) KCNH2HRH3HRH2HRH1KDM4E
Hydrochloric Acid SCHEMBL23247221 0.86 KDM4E (0.69) HRH2HRH1KDM4EALDH1A1MAPT
Hydrochloric Acid SCHEMBL8404070 0.86 KCNH2 (0.80) KCNH2HRH3HRH2HRH1KDM4E
SCHEMBL4441360 0.85 SMN1; SMN2 (0.73) KCNH2HRH3KDM4EALDH1A1MAPT
SCHEMBL20409779 0.83 LTA4H (0.64) KDM4EALDH1A1MAPTTDP1LTA4H
SCHEMBL4441264 0.82 HRH3 (0.61) KCNH2HRH3HRH2HRH1KDM4E
SCHEMBL15047632 0.82 KMT2A (0.63) HRH3HRH2HRH1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0435381-B1 Antipicornaviral pyridazinamines JANSSEN PHARMACEUTICA NV (BE) 1995-11-02 EP disclosed
EP-0398425-B1 Antirhinoviral piperidinyl, pyrrolidinyl and piperazinyl alkylphenol ethers JANSSEN PHARMACEUTICA NV (BE) 1994-03-16 EP disclosed
US-5196535-A Viricides JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-23 US disclosed
US-5100893-A Viricides, effective against picorna virus, durability JANSSEN PHARMACEUTICA N.V. (BE) 1992-03-31 US disclosed
EP-0435381-A1 Antipicornaviral pyridazinamines JANSSEN PHARMACEUTICA N.V. (BE) 1991-07-03 EP disclosed
EP-0398425-A1 Antirhinoviral piperidinyl, pyrrolidinyl and piperazinyl alkylphenol ethers JANSSEN PHARMACEUTICA N.V. (BE) 1990-11-22 EP disclosed