SCHEMBL5618488

SCHEMBL5618488

CC(C)NC(=O)NC(C)(C)CNc1c(N)cnc2cc(OCc3ccccc3)ccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN2 Q96KS0 2/20 0.41
EGLN1 Q9GZT9 2/20 0.41
MEN1 O00255 2/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 1/20 0.40
PTGES O14684 1/20 0.40
MAOA P21397 1/20 0.39
NMT1 P30419 2/20 0.39
PPARG P37231 2/20 0.38
MAOB P27338 1/20 0.37
MME P08473 1/20 0.37
ACE P12821 1/20 0.37
CPA1 P15085 1/20 0.37
ACE2 Q9BYF1 1/20 0.37
LTA4H P09960 1/20 0.37
KDR P35968 1/20 0.37
GPR132 Q9UNW8 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3873470 0.89 EGLN2 (0.44) EGLN2EGLN1MEN1MAPTKMT2A
SCHEMBL4069120 0.88 EGLN2 (0.43) EGLN2EGLN1MEN1MAPTKMT2A
SCHEMBL5618323 0.87 MAPT (0.40) EGLN2EGLN1MEN1MAPTKMT2A
SCHEMBL1486504 0.83 MAPT (0.42) EGLN2EGLN1MEN1MAPTKMT2A
SCHEMBL4066173 0.82 ALOX5 (0.40) EGLN2EGLN1MEN1MAPTKMT2A
SCHEMBL1486532 0.82 AR (0.40) EGLN2EGLN1MEN1MAPTKMT2A
SCHEMBL4070622 0.82 NMT1 (0.41) EGLN2EGLN1MEN1MAPTKMT2A
SCHEMBL3866418 0.82 NMT1 (0.48) EGLN2EGLN1MEN1MAPTKMT2A
SCHEMBL1486695 0.80 NMT1 (0.40) EGLN2EGLN1MEN1MAPTKMT2A
SCHEMBL1486517 0.79 MAPT (0.41) MEN1MAPTKMT2AMAOANMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9856254-B2 Alkoxy substituted imidazoquinolines 3M INNOVATIVE PROPERTIES COMPANY (US) 2018-01-02 US disclosed
US-20160280707-A1 ALKOXY SUBSTITUTED IMIDAZOQUINOLINES 3M INNOVATIVE PROPERTIES CO (US) 2016-09-29 US disclosed
US-9365567-B2 Alkoxy substituted imidazoquinolines 3M INNOVATIVE PROPERTIES COMPANY (US) 2016-06-14 US disclosed
US-8871782-B2 Alkoxy substituted imidazoquinolines 3M INNOVATIVE PROPERTIES COMPANY (US) 2014-10-28 US disclosed
US-20070060754-A1 Alkoxy substituted imidazoquinolines 3M INNOVATIVE PROPERTIES COMPANY 2007-03-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070060754-A1 Alkoxy substituted imidazoquinolines IL2, IFNG, IRF3 EGLN2 1301/4885EGLN1 1360/4885MEN1 3720/4885
US-20160280707-A1 ALKOXY SUBSTITUTED IMIDAZOQUINOLINES IL2, IFNG, IRF3 EGLN2 1301/4885EGLN1 1360/4885MEN1 3720/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.