SCHEMBL562256

SCHEMBL562256

CCCCCc1cc2c(nc(O)n2CC2CCOCC2)c(N(Cc2ccc(OC)cc2)Cc2ccc(OC)cc2)n1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.37
CYP2C19 P33261 2/20 0.37
HTR6 P50406 2/20 0.37
CNR2 P34972 9/20 0.36
CNR1 P21554 3/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2D6 P10635 2/20 0.35
HRH1 P35367 2/20 0.35
AVPR1B P47901 1/20 0.35
TLR7 Q9NYK1 1/20 0.34
RIPK3 Q9Y572 1/20 0.34
SLC2A1 P11166 1/20 0.34
CREBBP Q92793 1/20 0.33
P2RX3 P56373 1/20 0.33
PDE1B Q01064 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3339558 0.84 SLC2A1 (0.42) SLC2A1P2RX3
SCHEMBL562449 0.82 TLR7 (0.40) CNR2CYP2C9CYP2D6TLR7
SCHEMBL563383 0.82 TLR7 (0.45) TLR7
SCHEMBL562921 0.81 KCNH2 (0.41) KCNH2CYP2C9CYP2D6TLR7
SCHEMBL561914 0.78 TLR7 (0.39) CYP2C9CYP2D6TLR7
SCHEMBL562562 0.77 TLR7 (0.47) CNR2TLR7
SCHEMBL563312 0.75 DYRK1A (0.43) CNR2
SCHEMBL561529 0.75 TP53 (0.38) CYP2C9CYP2D6TLR7
SCHEMBL562667 0.70 TLR7 (0.43) CYP2C9CYP2D6TLR7
SCHEMBL563162 0.69 PTGS2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120035209-A1 Hydroxy Substituted 1H-Imidazopyridines and Methods PFIZER INC. (US) 2012-02-09 US disclosed
US-20100152230-A1 HYDROXY SUBSTITUTED 1H-IMIDAZOPYRIDINES AND METHODS PFIZER INC. 2010-06-17 US disclosed
EP-1924581-A1 HYDROXY SUBSTITUTED 1H-IMIDAZOPYRIDINES AND METHODS Pfizer, Inc. (US) 2008-05-28 EP disclosed
WO-2007028129-A1 HYDROXY SUBSTITUTED 1H-IMIDAZOPYRIDINES AND METHODS PFIZER INC. (US) 2007-03-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100152230-A1 HYDROXY SUBSTITUTED 1H-IMIDAZOPYRIDINES AND METHODS IL4, IL2, IL4I1 KCNH2 3737/4885CYP2C19 1913/4885HTR6 261/4885
US-20120035209-A1 Hydroxy Substituted 1H-Imidazopyridines and Methods IL2, IL4, IL4I1 KCNH2 3811/4885CYP2C19 2018/4885HTR6 286/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.