SCHEMBL5628181

SCHEMBL5628181

Oc1ccc(Cc2ccc(Br)cn2)cc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.46
ESR2 Q92731 4/20 0.46
LTC4S Q16873 1/20 0.44
ALOX15 P16050 1/20 0.43
MET P08581 1/20 0.41
AGER Q15109 1/20 0.41
MBOAT4 Q96T53 1/20 0.39
GBA1 P04062 1/20 0.38
EPHX2 P34913 1/20 0.38
KEAP1 Q14145 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17664387 0.81 KEAP1 (0.43) MBOAT4GBA1EPHX2KEAP1KDM4E
SCHEMBL17664018 0.81 GBA1 (0.48) MBOAT4GBA1EPHX2
SCHEMBL17663847 0.81 GBA1 (0.45) MBOAT4GBA1KDM4EALDH1A1
SCHEMBL16431630 0.80 ESR1 (0.59) ESR1ESR2METKEAP1
SCHEMBL5652510 0.78 ESR1 (0.46) ESR1ESR2ALOX15KEAP1KDM4E
SCHEMBL2250648 0.75 ESR1 (0.74) ESR1ESR2ALOX15AGERKEAP1
SCHEMBL28420432 0.75 CA2 (0.52)
SCHEMBL17664101 0.74 GBA1 (0.53) GBA1ALDH1A1
SCHEMBL1602934 0.73 ESR1 (0.47) ESR1ESR2ALDH1A1
SCHEMBL506458 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9765030-B2 Benzylamine derivatives and their utility as cholesterol ester-transfer protein inhibitors DR. REDDY'S LABORATORIES LTD. (IN) 2017-09-19 US disclosed
US-20140134235-A1 NOVEL BENZYLAMINE DERIVATIVES AND THEIR UTILITY AS CHOLESTEROL ESTER-TRANSFER PROTEIN INHIBITORS DR. REDDY'S LABORATORIES LTD. (IN) 2014-05-15 US disclosed
US-8604055-B2 Substituted benzylamino quinolines as cholesterol ester-transfer protein inhibitors DR. REDDY'S LABORATORIES LTD. (IN) 2013-12-10 US disclosed
US-20070015758-A1 Novel benzylamine derivatives and their utility as cholesterol ester-transfer protein inhibitors DR. REDDY'S LABORATORIES LTD. (IN) 2007-01-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140134235-A1 NOVEL BENZYLAMINE DERIVATIVES AND THEIR UTILITY AS CHOLESTEROL ESTER-TRANSFER PROTEIN INHIBITORS CETP, NPC1, DBI ESR1 4205/4885ESR2 2805/4885LTC4S 1393/4885
US-20070015758-A1 Novel benzylamine derivatives and their utility as cholesterol ester-transfer protein inhibitors CETP, NPC1, DBI ESR1 4205/4885ESR2 2805/4885LTC4S 1393/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.