Acetylcholine

Acetylcholine

SCHEMBL563048

CC(=O)OCC[N+](C)(C)C.N[C@@H](CCC(=O)O)C(=O)[O-]

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CHRM3

The experimentally established mechanism targets of Acetylcholine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 known ✓ P20309 8/20 0.54
CHRM1 P11229 8/20 0.54
CHRM2 P08172 7/20 0.54
CHRM4 P08173 7/20 0.54
CHRM5 P08912 6/20 0.54
CHRNB2 P17787 4/20 0.54
CHRNA4 P43681 4/20 0.54
CHRNA7 P36544 3/20 0.54
HTR1A P08908 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
PGR P06401 1/20 0.54
TBXA2R P21731 1/20 0.54
CHRNB4 P30926 1/20 0.54
CHRNA3 P32297 1/20 0.54
CHRNA10 Q9GZZ6 1/20 0.54
CHRNA9 Q9UGM1 1/20 0.54
GALR3 O60755 2/20 0.53
GAA P10253 1/20 0.53
RAB9A P51151 1/20 0.53
ADRA2A P08913 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetylcholine SCHEMBL563047 0.90 CHRM1 (0.56) CHRM1CHRM3CHRM2CHRM4CHRM5
Acetylcholine SCHEMBL28345020 0.88 CHRM1 (0.58) CHRM1CHRM3CHRM2CHRM4CHRM5
Acetylcholine SCHEMBL17629404 0.85 CHRM1 (0.58) CHRM1CHRM3CHRM2CHRM4CHRM5
SCHEMBL8218840 0.82 ADRA2A (0.50) CHRM1CHRM3CHRM2CHRM4CHRM5
Acetylcholine SCHEMBL17629405 0.81 CHRM1 (0.59) CHRM1CHRM3CHRM2CHRM4CHRM5
Acetylcholine SCHEMBL17629403 0.81 CHRM1 (0.59) CHRM1CHRM3CHRM2CHRM4CHRM5
D-Glutamate SCHEMBL8218834 0.80 CYP1A2 (0.46) CYP2C19LMNAMAPTBLMTSHR
Acetylcholine SCHEMBL29441892 0.80 CHRM1 (0.68) CHRM1CHRM3CHRM2CHRM4CHRM5
Acetylcholine SCHEMBL28054287 0.78 CHRM1 (0.83) CHRM1CHRM3CHRM2CHRM4CHRM5
D-Glutamate SCHEMBL2208071 0.77 TSHR (0.50) CYP2C19LMNAMAPTBLMTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070287991-A1 Devices and methods for detection of markers of axial pain with or without radiculopathy MEDTRONIC, INC. 2007-12-13 US claimed
US-9675657-B2 Role of an herbal formulation in the prevention and management of age related neurodegenerative disorders with special reference to senile dementia SRM UNIVERSITY (IN) 2017-06-13 US disclosed
EP-1634075-B1 Electronic device for communication with living cells YISSUM RES DEV CO (IL) 2015-01-14 EP disclosed
WO-2012020423-A1 ROLE OF AN HERBAL FORMULATION IN THE PREVENTION AND MANAGEMENT OF AGE RELATED NEURODEGENERATIVE DISORDERS WITH SPECIAL REFERENCE TO SENILE DEMENTIA INTERDISCIPLINARY SCHOOL OF INDIAN SYSTEM OF MEDICINE (IN) 2012-02-16 WO disclosed
US-20120034324-A1 ROLE OF AN HERBAL FORMULATION IN THE PREVENTION AND MANAGEMENT OF AGE RELATED NEURODEGENERATIVE DISORDERS WITH SPECIAL REFERENCE TO SENILE DEMENTIA SRM UNIVERSITY (IN) 2012-02-09 US disclosed
US-7795039-B2 provides a surface-substrate for adherence of cells; comprises a micronail structure protruding from the surface, a region of the micronail having cellular-internalization promoting properties; for research purposes, for photography purposes; provide a good electrical and/or chemical coupling YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2010-09-14 US disclosed
US-20070099173-A1 provides a surface-substrate for adherence of cells; comprises a micronail structure protruding from the surface, a region of the micronail having cellular-internalization promoting properties; for research purposes, for photography purposes; provide a good electrical and/or chemical coupling YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2007-05-03 US disclosed
EP-1634075-A1 ELECTRONIC DEVICE FOR COMMUNICATION WITH LIVING CELLS YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2006-03-15 EP disclosed
WO-2004109282-A1 ELECTRONIC DEVICE FOR COMMUNICATION WITH LIVING CELLS YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2004-12-16 WO disclosed