SCHEMBL5632392

SCHEMBL5632392

CCC[CH]c1ccc(C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.42
CYP1A2 P05177 1/20 0.41
AHR P35869 1/20 0.40
NQO2 P16083 2/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA7 P36544 1/20 0.40
CHRNA4 P43681 1/20 0.40
PTGS2 P35354 1/20 0.40
CYP1A1 P04798 2/20 0.39
CYP1B1 Q16678 2/20 0.39
FBP1 P09467 1/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
HDAC3 O15379 1/20 0.38
ADAM17 P78536 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1992348 0.85 PTGS1 (0.46) PTGS1CYP1A2AHRNQO2CHRNB2
SCHEMBL18242615 0.84 NR1H2 (0.33) PTGS1
SCHEMBL5358981 0.82 ALDH1A1 (0.37) MEN1KMT2A
SCHEMBL18242019 0.81 NR1H2 (0.32)
SCHEMBL1611685 0.81 CYP1A2 (0.42) CYP1A2CA1CA2HDAC3HDAC1
SCHEMBL28202493 0.81 KDM1A (0.45) CA1CA2HDAC1MAOB
SCHEMBL7019012 0.80 CYP1A2 (0.47) PTGS1CYP1A2AHRNQO2CHRNB2
SCHEMBL22483309 0.80 CYP1A2 (0.47) PTGS1CYP1A2AHRNQO2CHRNB2
SCHEMBL18378569 0.80 NR1H2 (0.31)
SCHEMBL11659879 0.79 AHR (0.44) PTGS1CYP1A2AHRNQO2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10451967-B2 Acid- and radical-generating agent and method for generating acid and radical FUJIFILM WAKO PURE CHEMICAL CORPORATION (JP) 2019-10-22 US disclosed
US-20160342084-A1 ACID- AND RADICAL-GENERATING AGENT AND METHOD FOR GENERATING ACID AND RADICAL FUJIFILM WAKO PURE CHEMICAL CORPORATION (JP) 2016-11-24 US disclosed
US-20070232678-A1 (4, 5, 6, 7-Tetrahydro-1-H-Indol-7-Yl) Acetic Acid Derivatives for Treatment of Alzheimer's Disease MERCK SHARP & DOHME LTD. (GB) 2007-10-04 US disclosed
US-4740332-A HYPOPHOSPHORUS ACID OR SALT WITH ALPHA OLEFINS E. R. SQUIBB & SONS, INC. (US) 1988-04-26 US disclosed
EP-0246015-A2 Process for preparing phosphonous acids E.R. Squibb & Sons, Inc. (US) 1987-11-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070232678-A1 (4, 5, 6, 7-Tetrahydro-1-H-Indol-7-Yl) Acetic Acid Derivatives for Treatment of Alzheimer's Disease APP, BACE1, CHAT PTGS1 791/4885CYP1A2 572/4885AHR 167/4885
US-10451967-B2 Acid- and radical-generating agent and method for generating acid and radical CBR1, HAO2, CBR3 PTGS1 758/4885CYP1A2 360/4885AHR 159/4885
US-20160342084-A1 ACID- AND RADICAL-GENERATING AGENT AND METHOD FOR GENERATING ACID AND RADICAL CBR1, HAO2, CBR3 PTGS1 758/4885CYP1A2 360/4885AHR 159/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.