Brivaracetam

Brivaracetam

SCHEMBL563380

CCCC1CC(=O)N([C@@H](CC)C(N)=O)C1

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SV2A

The experimentally established mechanism targets of Brivaracetam. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
LMNA P02545 1/20 0.49
CA12 O43570 1/20 0.49
CA3 P07451 1/20 0.49
CA4 P22748 1/20 0.49
CA6 P23280 1/20 0.49
CA5A P35218 1/20 0.49
CA7 P43166 1/20 0.49
CA9 Q16790 1/20 0.49
CA13 Q8N1Q1 1/20 0.49
CA14 Q9ULX7 1/20 0.49
CA5B Q9Y2D0 1/20 0.49
BRD4 O60885 3/20 0.38
MAPT P10636 2/20 0.35
TSHR P16473 1/20 0.33
CYP2C9 P11712 1/20 0.33
ALDH1A1 P00352 1/20 0.32
APEX1 P27695 1/20 0.31
BLM P54132 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Brivaracetam SCHEMBL22446812 1.00 CA1 (0.49) CA1CA2LMNACA12CA3
Brivaracetam SCHEMBL13596590 1.00 CA1 (0.49) CA1CA2LMNACA12CA3
Brivaracetam SCHEMBL563918 1.00 CA1 (0.49) CA1CA2LMNACA12CA3
Brivaracetam SCHEMBL563970 1.00 CA1 (0.49) CA1CA2LMNACA12CA3
Brivaracetam SCHEMBL122081 1.00 CA1 (0.49) CA1CA2LMNACA12CA3
Brivaracetam SCHEMBL564055 1.00 CA1 (0.49) CA1CA2LMNACA12CA3
Brivaracetam SCHEMBL2408675 1.00 CA1 (0.49) CA1CA2LMNACA12CA3
Brivaracetam SCHEMBL563666 1.00 CA1 (0.49) CA1CA2LMNACA12CA3
SCHEMBL563677 0.93 LMNA (0.41) CA1CA2LMNACA12CA3
SCHEMBL563118 0.91 LMNA (0.40) CA1CA2LMNACA12CA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 97 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8642641-B2 Co-crystals of pyrrolidinones UCB PHARMA, S.A. (BE) 2014-02-04 US claimed
EP-2041084-B1 CO-CRYSTALS OF PYRROLIDINONES UCB PHARMA SA (BE) 2013-11-06 EP claimed
US-20120245215-A1 Co-Crystals of Pyrrolidinones UCB PHARMA, S.A. (BE) 2012-09-27 US claimed
US-20100240728-A1 Co-Crystals of Pyrrolidinones UCB PHARMA, S.A. (BE) 2010-09-23 US claimed
EP-1452524-B1 \"2-oxo-1-pyrrolidine derivative and its pharmaceutical uses\ UCB PHARMA SA (BE) 2009-10-14 EP claimed
CN-101506157-A Co-crystals of pyrrolidinones UCB PHARMA SA (BE) 2009-08-12 CN claimed
EP-2041084-A1 CO-CRYSTALS OF PYRROLIDINONES UCB Pharma, S.A. (BE) 2009-04-01 EP claimed
WO-2007141002-A1 CO-CRYSTALS OF PYRROLIDINONES UCB PHARMA, S.A. (BE) 2007-12-13 WO claimed
US-6911461-B2 For treating epilepsy, epileptogenesis, seizure disorders, convulsions, bipolar disorders, mania, depression, anxiety, migraine, neuralgia, chronic pain, neuropathic pain, cerebral ischemia, cardiac arrhythmia, myotonia, cocaine abuse UCB, S.A. (BE) 2005-06-28 US claimed
EP-1452524-A1 \"2-oxo-1-pyrrolidine derivative and its pharmaceutical uses\ UCB, S.A. (BE) 2004-09-01 EP claimed
US-20040116507-A1 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses UCB Biopharma SRL (BE) 2004-06-17 US claimed
US-20030120080-A1 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses UCB Biopharma SRL (BE) 2003-06-26 US claimed
EP-1265862-A2 2-OXO-1-PYRROLIDINE DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB, S.A. (BE) 2002-12-18 EP claimed
WO-2001062726-A2 2-OXO-1-PYRROLIDINE DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB, S.A. (BE) 2001-08-30 WO claimed
CN-117466797-A Preparation method of Brivaracetam 重庆普佑生物医药有限公司 2024-01-30 CN disclosed
CN-117447374-A New method for preparing brivaracetam 重庆普佑生物医药有限公司 2024-01-26 CN disclosed
EP-3302441-B1 PROCESSES TO PRODUCE BRIVARACETAM SUZHOU PENGXU PHARMATECH CO LTD (CN) 2023-12-13 EP disclosed
US-20030120080-A1 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses UCB Biopharma SRL (BE) 2003-06-26 US disclosed
EP-1265862-A2 2-OXO-1-PYRROLIDINE DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB, S.A. (BE) 2002-12-18 EP disclosed
WO-2001062726-A2 2-OXO-1-PYRROLIDINE DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB, S.A. (BE) 2001-08-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120245215-A1 Co-Crystals of Pyrrolidinones PYCR1, CCNT1, PRMT1 CA1 1299/4885CA2 2448/4885LMNA 3002/4885
US-20030120080-A1 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses CYP1B1, CYP1A2, OGDH CA1 1842/4885CA2 1417/4885LMNA 3771/4885
US-20100240728-A1 Co-Crystals of Pyrrolidinones PYCR1, C1S, CCNT1 CA1 1434/4885CA2 2766/4885LMNA 2662/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.