SCHEMBL5634675

SCHEMBL5634675

CS(=O)(=O)Nc1ccc(Cc2noc(C3CCN(CC[C@H](NC(=O)CC(F)(F)F)c4ccccc4)CC3)n2)cc1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 11/20 0.46
PRCP P42785 5/20 0.40
CCR2 P41597 1/20 0.39
CYP2D6 P10635 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5633684 0.91 CCR5 (0.51) CCR5PRCPCYP2D6OPRM1OPRD1
SCHEMBL5633692 0.91 CCR5 (0.51) CCR5PRCPCYP2D6OPRM1OPRD1
SCHEMBL5634122 0.90 CCR5 (0.47) CCR5PRCPCYP2D6OPRM1OPRD1
SCHEMBL5635080 0.89 CCR5 (0.49) CCR5PRCPCCR2KCNH2
SCHEMBL5633870 0.88 CCR5 (0.60) CCR5KCNH2
SCHEMBL14514104 0.87 CCR5 (0.46) CCR5PRCPCYP2D6OPRM1OPRD1
SCHEMBL5633685 0.86 CCR5 (0.54) CCR5KCNH2
SCHEMBL5633851 0.85 CCR5 (0.52) CCR5PRCPKCNH2
SCHEMBL14514107 0.83 CCR5 (0.43) CCR5PRCPCYP2D6OPRM1OPRD1
Hydrochloric Acid SCHEMBL5634554 0.83 CCR5 (0.42) CCR5PRCPCYP2D6OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US claimed
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US disclosed
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US disclosed
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US disclosed
US-20010039026-A1 Assay method PFIZER INC. 2001-11-08 US disclosed
EP-1118858-A2 Assay method Pfizer Limited (GB) 2001-07-25 EP disclosed