SCHEMBL5634879

SCHEMBL5634879

O=C(N[C@@H](CCN1CCC(c2nc(Cc3ccc(F)cc3)no2)CC1)c1ccccc1)C1CCOCC1

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.58
KCNH2 Q12809 1/20 0.47
PRCP P42785 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5661678 0.94 CCR5 (0.65) CCR5KCNH2
SCHEMBL5635173 0.94 CCR5 (0.65) CCR5KCNH2
SCHEMBL5633916 0.90 CCR5 (0.53) CCR5KCNH2PRCP
SCHEMBL5633911 0.90 CCR5 (0.53) CCR5KCNH2PRCP
SCHEMBL5634369 0.89 CCR5 (0.73) CCR5KCNH2
SCHEMBL5635539 0.89 CCR5 (0.73) CCR5KCNH2
SCHEMBL5634413 0.88 CCR5 (0.64) CCR5KCNH2
SCHEMBL5633685 0.88 CCR5 (0.54) CCR5KCNH2
SCHEMBL5634195 0.87 CCR5 (0.67) CCR5KCNH2
SCHEMBL14514138 0.87 CCR5 (0.65) CCR5KCNH2PRCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US claimed
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US disclosed
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US disclosed
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US disclosed
US-20010039026-A1 Assay method PFIZER INC. 2001-11-08 US disclosed
EP-1118858-A2 Assay method Pfizer Limited (GB) 2001-07-25 EP disclosed