SCHEMBL5638181

SCHEMBL5638181

CC(C)(C)OC(=O)N1CCc2c(c3c(-c4ccc(Cl)c(Cl)c4)ccc4c3n2CCCS4)C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.37
CYBB P04839 1/20 0.36
NOX5 Q96PH1 1/20 0.36
NOX4 Q9NPH5 1/20 0.36
NOX1 Q9Y5S8 1/20 0.36
NR1H2 P55055 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MKNK1 Q9BUB5 3/20 0.33
KDM1A O60341 1/20 0.33
PRKCZ Q05513 1/20 0.32
RORC P51449 2/20 0.32
RET P07949 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5636457 0.85 CYBB (0.38) ESR2CYBBNOX5NOX4NOX1
SCHEMBL5637696 0.85 GPR119 (0.38) ESR2CYBBNOX5NOX4NOX1
SCHEMBL5635040 0.82 ESR2 (0.38) ESR2CYBBNOX5NOX4NOX1
SCHEMBL5636204 0.82 ESR2 (0.38) ESR2CYBBNOX5NOX4NOX1
SCHEMBL5507669 0.70 PTGDR2 (0.39) ALDH1A1LMNAMAPTHPGDSMN1; SMN2
SCHEMBL8355563 0.70 ESR2 (0.53) ESR2NR1H2MEN1KMT2AMKNK1
SCHEMBL4791213 0.66 ESR2 (0.44) ESR2CYBBNOX5NOX4NOX1
SCHEMBL3184176 0.65 ESR2 (0.47) ESR2NR1H2MAPTMEN1KMT2A
SCHEMBL3194232 0.64 SLC6A3 (0.57) ESR2NR1H2
SCHEMBL28443721 0.64 STS (0.45) ESR2CYBBNOX5NOX4NOX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed