SCHEMBL5645453

SCHEMBL5645453

N#Cc1ccc(Nc2ccccc2)c(Br)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.66
KDM4E B2RXH2 3/20 0.66
GAA P10253 3/20 0.66
CXCR2 P25025 5/20 0.51
CXCR1 P25024 2/20 0.47
MAPT P10636 3/20 0.46
HTT P42858 3/20 0.46
MEN1 O00255 2/20 0.46
LMNA P02545 2/20 0.46
KMT2A Q03164 2/20 0.46
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ABCG2 Q9UNQ0 4/20 0.44
ABCB1 P08183 3/20 0.44
GSK3B P49841 2/20 0.41
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
CSNK1A1 P48729 1/20 0.40
CSNK1D P48730 1/20 0.40
CSNK1G2 P78368 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16197958 0.84 KDM4E (0.72) ALDH1A1KDM4EGAACXCR2CXCR1
SCHEMBL28248993 0.81 KDM4E (0.68) ALDH1A1KDM4EGAACXCR2CXCR1
SCHEMBL13610402 0.79 GAA (1.00) ALDH1A1KDM4EGAACXCR2CXCR1
SCHEMBL29642859 0.79 GAA (1.00) ALDH1A1KDM4EGAACXCR2CXCR1
SCHEMBL13750111 0.78 ALDH1A1 (0.69) ALDH1A1KDM4EGAACXCR2CXCR1
SCHEMBL18796197 0.77 ALPL (0.48) ALDH1A1KDM4EGAACXCR2HTT
SCHEMBL24524348 0.76 GAA (0.61) ALDH1A1KDM4EGAACXCR2CXCR1
SCHEMBL11900810 0.76 GAA (0.76) ALDH1A1KDM4EGAACXCR2CXCR1
SCHEMBL14428159 0.76 ALK (0.51) ALDH1A1KDM4EGAAMAPTHTT
SCHEMBL28598854 0.76 ALDH1A1 (0.54) ALDH1A1KDM4EGAAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8343981-B2 Heterocyclyl-substituted dihydroquinazolines and their use as antiviral agents AICURIS GMBH & CO. KG (DE) 2013-01-01 US disclosed
US-20070185121-A1 Heterocyclyl-substituted dihydroquinazolines and their use as antiviral agents BAYER HEALTHCARE AG (DE) 2007-08-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070185121-A1 Heterocyclyl-substituted dihydroquinazolines and their use as antiviral agents TYMP, RPL35, EIF2AK2 ALDH1A1 1660/4885KDM4E 2609/4885GAA 232/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.