SCHEMBL5650019

SCHEMBL5650019

COCCOc1cc2[nH]ccc(=O)c2cc1OC

nearest known ligand 0.75

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 1/20 0.48
KDM4E B2RXH2 3/20 0.43
MAPK1 P28482 1/20 0.43
ALDH1A1 P00352 4/20 0.40
HSD17B10 Q99714 1/20 0.40
KDR P35968 9/20 0.40
MAPT P10636 2/20 0.40
HPGD P15428 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CTSV O60911 1/20 0.38
CTSL P07711 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29842783 0.89 IMPDH2 (0.48) IMPDH2KDM4EMAPK1ALDH1A1HSD17B10
SCHEMBL16207483 0.89 IMPDH2 (0.48) IMPDH2KDM4EMAPK1ALDH1A1HSD17B10
SCHEMBL7291390 0.88 PDE3B (0.51) IMPDH2KDM4EMAPK1ALDH1A1MAPT
SCHEMBL7294056 0.87 IMPDH2 (0.49) IMPDH2KDM4EMAPK1ALDH1A1HSD17B10
SCHEMBL372048 0.87 IMPDH2 (0.58) IMPDH2KDM4EALDH1A1HSD17B10MAPT
SCHEMBL7284981 0.86 IMPDH2 (0.50) IMPDH2KDM4EMAPK1ALDH1A1HSD17B10
SCHEMBL7290454 0.86 IMPDH2 (0.50) IMPDH2KDM4EMAPK1ALDH1A1HSD17B10
SCHEMBL15275124 0.86 IMPDH2 (0.50) IMPDH2KDM4EMAPK1ALDH1A1HSD17B10
SCHEMBL1892646 0.82 PRKCQ (0.40) IMPDH2ALDH1A1
SCHEMBL1894760 0.82 PRKAB2 (0.49) IMPDH2KDM4EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0343574-B1 4(1H)-quinolone derivatives KIRIN BREWERY (JP) 1994-07-27 EP claimed
US-20070299092-A1 Quinone Substituted Quinazoline and Quinoline Kinase Inhibitors WYETH (US) 2007-12-27 US disclosed
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP disclosed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US disclosed
EP-0343574-B1 4(1H)-quinolone derivatives KIRIN BREWERY (JP) 1994-07-27 EP disclosed
US-5081121-A Cardiotonic agents KIRIN BEER KABUSHIKI KAISHA (JP) 1992-01-14 US disclosed
EP-0343574-A1 4(1H)-quinolone derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1989-11-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070299092-A1 Quinone Substituted Quinazoline and Quinoline Kinase Inhibitors KDR, FLT1, FLT4 IMPDH2 2971/4885KDM4E 1380/4885MAPK1 139/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.