SCHEMBL5654192

SCHEMBL5654192

CCC(O)C(C)N(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.55
HPGD P15428 1/20 0.44
SIGMAR1 Q99720 1/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
TSHR P16473 3/20 0.42
ALDH1A1 P00352 1/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
CA12 O43570 2/20 0.42
CA9 Q16790 2/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
SLC6A2 P23975 1/20 0.42
HTR2A P28223 1/20 0.42
SLC6A4 P31645 1/20 0.42
ADRA1A P35348 1/20 0.42
OPRK1 P41145 1/20 0.42
SLC6A3 Q01959 1/20 0.42
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8950842 0.84 TSHR (0.44) TRPA1HPGDSIGMAR1KMT2AMEN1
SCHEMBL14541169 0.84 TSHR (0.44) TRPA1HPGDSIGMAR1KMT2AMEN1
SCHEMBL8950839 0.84 TSHR (0.44) TRPA1HPGDSIGMAR1KMT2AMEN1
SCHEMBL5889904 0.82 TRPA1 (0.41) TRPA1HPGDSIGMAR1KMT2AMEN1
SCHEMBL26989268 0.82 TSHR (0.46) TRPA1HPGDSIGMAR1KMT2AMEN1
SCHEMBL26988083 0.82 TSHR (0.46) TRPA1HPGDSIGMAR1KMT2AMEN1
SCHEMBL26987985 0.82 TSHR (0.46) TRPA1HPGDSIGMAR1KMT2AMEN1
SCHEMBL26988540 0.82 TSHR (0.46) TRPA1HPGDSIGMAR1KMT2AMEN1
SCHEMBL428101 0.82 TSHR (0.46) TRPA1HPGDSIGMAR1KMT2AMEN1
SCHEMBL29929713 0.82 TRPA1 (0.51) TRPA1HPGDSIGMAR1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235082-A1 Long-chain, straight-chain 2-amino-3-hydroxyalkanes RINEHART KENNETH L 2006-10-19 US disclosed
US-7109244-B2 Compositions and methods comprising long-chain, straight-chain 2-amino-3-hydroxyalkanes RINEHART KENNETH L 2006-09-19 US disclosed
US-20060183806-A9 COMPOSITIONS AND METHODS COMPRISING LONG-CHAIN, STRAIGHT-CHAIN 2-AMINO-3- HYDROXYALKANES RINEHART KENNETH L 2006-08-17 US disclosed
US-RE38793-E1 Spisulosine compounds RINEHART KENNETH L 2005-09-06 US disclosed
EP-1069894-B1 SPISULOSINE COMPOUNDS HAVING ANTITUMOUR ACTIVITY UNIV ILLINOIS (US) 2005-08-31 EP disclosed
US-6800661-B1 Spisulosine compounds BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2004-10-05 US disclosed
US-20040147615-A1 Spisulosine compounds RINEHART KENNETH L (US) 2004-07-29 US disclosed
EP-1069894-A1 SPISULOSINE COMPOUNDS HAVING ANTITUMOUR ACTIVITY The Board of Trustees for the University of Illinois (US) 2001-01-24 EP disclosed
US-6107520-A SHOW UNIQUE CYTOTOXICITY AGAINST MURINE LYMPHOCYTIC LEUKEMIA CELLS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2000-08-22 US disclosed
WO-1999052521-A1 SPISULOSINE COMPOUNDS HAVING ANTITUMOUR ACTIVITY THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 1999-10-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060235082-A1 Long-chain, straight-chain 2-amino-3-hydroxyalkanes SLC3A2, HACL2, CLSPN TRPA1 489/4885HPGD 1344/4885SIGMAR1 309/4885
US-20040147615-A1 Spisulosine compounds CLSPN, SPIN3, OAT TRPA1 1152/4885HPGD 2908/4885SIGMAR1 616/4885
US-20060183806-A9 COMPOSITIONS AND METHODS COMPRISING LONG-CHAIN, STRAIGHT-CHAIN 2-AMINO-3- HYDROXYALKANES NEFM, OAT, POLM TRPA1 2074/4885HPGD 1239/4885SIGMAR1 571/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.