SCHEMBL5656069

SCHEMBL5656069

CCCn1ccnc1CO

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
POLB P06746 1/20 0.44
KMT2A Q03164 1/20 0.44
TLR8 Q9NR97 2/20 0.42
KCNH2 Q12809 1/20 0.39
HTT P42858 1/20 0.37
PDE4A P27815 2/20 0.36
PDE1A P54750 2/20 0.36
PDE1B Q01064 2/20 0.36
PDE4B Q07343 2/20 0.36
PDE4C Q08493 2/20 0.36
PDE4D Q08499 2/20 0.36
PDE1C Q14123 2/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
ALPG P10696 2/20 0.35
PLAA Q9Y263 1/20 0.35
FDPS P14324 1/20 0.34
ALPL P05186 1/20 0.34
AGTR1 P30556 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5655366 0.89 ALDH1A1 (0.59) ALDH1A1POLBKMT2ATLR8KCNH2
SCHEMBL5655435 0.87 TLR8 (0.59) ALDH1A1POLBKMT2ATLR8KCNH2
SCHEMBL2647561 0.83
SCHEMBL17865370 0.83 KCNH2 (0.41) ALDH1A1POLBKMT2ATLR8KCNH2
SCHEMBL4233920 0.83 TLR8 (0.48) ALDH1A1POLBKMT2ATLR8KCNH2
Hydrochloric Acid SCHEMBL1187702 0.82 KMT2A (0.42) ALDH1A1POLBKMT2ATLR8KCNH2
SCHEMBL4227889 0.82 ALDH1A1 (0.46) ALDH1A1POLBKMT2ATLR8KCNH2
Bromide SCHEMBL28149514 0.82 TLR8 (0.47) ALDH1A1POLBKMT2ATLR8KCNH2
SCHEMBL22710048 0.80 TLR8 (0.46) ALDH1A1POLBKMT2ATLR8KCNH2
SCHEMBL8026054 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7262185-B2 Benzazepine derivative, process for producing the same, and use TAKEDA CHEMICAL INDUSTRIES LTD. (JP) 2007-08-28 US disclosed
US-20040235822-A1 Benzazepine derivative, process for producing the same, and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-11-25 US disclosed
EP-1422228-A1 BENZAZEPINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE Takeda Chemical Industries, Ltd. (JP) 2004-05-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040235822-A1 Benzazepine derivative, process for producing the same, and use CYP1B1, CYP1A1, CYP2E1 ALDH1A1 519/4885POLB 3578/4885KMT2A 391/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.