SCHEMBL17865370

SCHEMBL17865370

OCCn1ccnc1CO

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.41
ALDH1A1 P00352 3/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 2/20 0.34
POLB P06746 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
FPR2 P25090 1/20 0.34
ALPG P10696 2/20 0.33
PLAA Q9Y263 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
ALPL P05186 1/20 0.33
FDPS P14324 1/20 0.33
TLR8 Q9NR97 2/20 0.32
LMNA P02545 2/20 0.32
MEN1 O00255 1/20 0.32
ADORA2B P29275 1/20 0.32
ESR1 P03372 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20425451 0.85 KCNH2 (0.42) KCNH2CCNE1CDK2FPR2ALPG
SCHEMBL26196840 0.83 ALPG (0.48) KCNH2ALDH1A1KMT2APOLBFPR2
Bromide SCHEMBL18979889 0.83 KCNH2 (0.41) KCNH2CCNE1CDK2FPR2ALPG
SCHEMBL23053790 0.83 KCNH2 (0.33) KCNH2ALDH1A1KMT2APOLBCCNE1
SCHEMBL5656069 0.83 ALDH1A1 (0.44) KCNH2ALDH1A1HTTKMT2APOLB
SCHEMBL8026054 0.82
SCHEMBL11295344 0.80 KCNH2 (0.42) KCNH2ALDH1A1KMT2APOLBALPG
SCHEMBL5655366 0.80 ALDH1A1 (0.59) KCNH2ALDH1A1HTTKMT2APOLB
SCHEMBL14416076 0.80 TLR8 (0.40) KCNH2ALDH1A1HTTKMT2APOLB
Bromide SCHEMBL28684914 0.80 AGTR1 (0.35) KCNH2ALDH1A1KMT2APOLBALPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10108129-B2 Member for electrophotography and method of producing the member, process cartridge, and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2018-10-23 US claimed
US-20160187809-A1 MEMBER FOR ELECTROPHOTOGRAPHY AND METHOD OF PRODUCING THE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2016-06-30 US claimed
EP-3037889-A1 MEMBER FOR ELECTROPHOTOGRAPHY AND METHOD OF PRODUCING THE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS Canon Kabushiki Kaisha (JP) 2016-06-29 EP claimed
EP-3037889-B1 MEMBER FOR ELECTROPHOTOGRAPHY AND METHOD OF PRODUCING THE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KK (JP) 2023-11-29 EP disclosed
US-10108129-B2 Member for electrophotography and method of producing the member, process cartridge, and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2018-10-23 US disclosed
EP-2970254-B1 IMIDAZO PYRIDINE COMPOUNDS LILLY CO ELI (US) 2017-06-21 EP disclosed
US-20160187809-A1 MEMBER FOR ELECTROPHOTOGRAPHY AND METHOD OF PRODUCING THE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2016-06-30 US disclosed
EP-3037889-A1 MEMBER FOR ELECTROPHOTOGRAPHY AND METHOD OF PRODUCING THE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS Canon Kabushiki Kaisha (JP) 2016-06-29 EP disclosed