SCHEMBL5658556

SCHEMBL5658556

Cc1ccc(OC(=O)COc2ncc(C(=O)Nc3ccc(F)cc3)cn2)c(C)c1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
MAPT P10636 2/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
CXCR1 P25024 10/20 0.52
CXCR2 P25025 10/20 0.52
ALDH1A1 P00352 1/20 0.48
RECQL P46063 1/20 0.44
F2 P00734 1/20 0.44
P4HTM Q9NXG6 1/20 0.44
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5658828 0.84 CXCR1 (0.51) NPC1RAB9ASMN1; SMN2CXCR1CXCR2
SCHEMBL5661096 0.84 CXCR2 (0.67) NPC1RAB9ASMN1; SMN2MAPTCXCR1
SCHEMBL5658045 0.82 CXCR2 (0.59) NPC1RAB9AMEN1KMT2ACXCR1
SCHEMBL5658349 0.81 CXCR2 (0.73) NPC1RAB9ACXCR1CXCR2ALDH1A1
SCHEMBL5656795 0.81 CXCR2 (0.76) NPC1RAB9ASMN1; SMN2MAPTMEN1
SCHEMBL5656391 0.80 CXCR1 (0.75) MAPTMEN1KMT2ACXCR1CXCR2
SCHEMBL5659069 0.80 CXCR2 (0.59) NPC1RAB9AMAPTCXCR1CXCR2
SCHEMBL5660773 0.80 CXCR2 (0.52) KMT2ACXCR1CXCR2ALDH1A1RECQL
SCHEMBL5660902 0.77 CXCR1 (0.56) NPC1RAB9ASMN1; SMN2CXCR1CXCR2
SCHEMBL5662987 0.77 CXCR2 (0.51) NPC1RAB9ASMN1; SMN2MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176310-B1 Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents UCB SA (GB) 2007-02-13 US disclosed