SCHEMBL5659183

SCHEMBL5659183

NC(=O)N1CCCN(C2CCN(C(=O)[CH]Cc3ccc4[nH]ncc4c3)CC2)CC1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 6/20 0.44
CYP3A4 P08684 6/20 0.44
ACACB O00763 4/20 0.41
ACACA Q13085 4/20 0.41
ROCK2 O75116 9/20 0.39
RPS6KB1 P23443 1/20 0.38
CLK2 P49760 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
STK17A Q9UEE5 1/20 0.38
DDR1 Q08345 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5661005 1.00 CALCRL (0.44) CALCRLCYP3A4ACACBACACAROCK2
SCHEMBL5661183 0.96 ACACB (0.42) CALCRLCYP3A4ACACBACACAROCK2
SCHEMBL5659149 0.96 ACACB (0.42) CALCRLCYP3A4ACACBACACAROCK2
SCHEMBL5660671 0.87 ROCK2 (0.44) CYP3A4ROCK2
SCHEMBL5658597 0.84 CALCA (0.48) CALCRL
SCHEMBL5658244 0.84 CALCA (0.48) CALCRL
SCHEMBL5660300 0.81 CCR3 (0.47) CALCRLCYP3A4ACACBACACA
SCHEMBL5660912 0.81 CCR3 (0.47) CALCRLCYP3A4ACACBACACA
SCHEMBL5659618 0.81 ACACB (0.37) CALCRLCYP3A4ACACBACACA
SCHEMBL5661224 0.81 ACACB (0.37) CALCRLCYP3A4ACACBACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227968-A1 Selected CGRP-antagonists process for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-10-13 US claimed
US-7205294-B2 Selected CGRP-antagonists process for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-04-17 US disclosed
US-20050227968-A1 Selected CGRP-antagonists process for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-10-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050227968-A1 Selected CGRP-antagonists process for preparing them and their use as pharmaceutical compositions BDKRB1, BDKRB2, CALCRL CALCRL 3/4885CYP3A4 1053/4885ACACB 4648/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.