SCHEMBL5659538

SCHEMBL5659538

Nc1nc(SCC(=O)O)ncc1C(=O)Nc1ccc(F)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 3/20 0.56
PTPN11 Q06124 1/20 0.48
RAB9A P51151 2/20 0.48
POLB P06746 1/20 0.48
PDE4B Q07343 1/20 0.47
LMNA P02545 5/20 0.47
MAPT P10636 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
SMN1; SMN2 Q16637 4/20 0.46
HTT P42858 2/20 0.46
HSD17B10 Q99714 2/20 0.46
TP53 P04637 1/20 0.46
GAA P10253 1/20 0.46
ALOX15 P16050 1/20 0.46
CXCR1 P25024 1/20 0.45
ATR Q13535 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5660105 0.87 CXCR1 (0.58) CXCR2PTPN11PDE4BLMNAMAPT
SCHEMBL5657757 0.85 ALDH1A1 (0.58) CXCR2PTPN11RAB9ALMNAMAPT
SCHEMBL5660845 0.84 CXCR1 (0.47) CXCR2PTPN11RAB9APDE4BLMNA
SCHEMBL5657939 0.83 CXCR2 (0.53) CXCR2RAB9APOLBLMNAMAPT
SCHEMBL5658940 0.83 LMNA (0.45) CXCR2PTPN11RAB9APDE4BLMNA
SCHEMBL5659631 0.83 CXCR1 (0.62) CXCR2PTPN11RAB9ALMNAMAPT
SCHEMBL5658611 0.82 CXCR1 (0.46) CXCR2PTPN11RAB9APDE4BLMNA
SCHEMBL5657961 0.82 SMN1; SMN2 (0.49) CXCR2RAB9ALMNAMAPTMEN1
SCHEMBL5659975 0.81 CXCR2 (0.73) CXCR2RAB9ACXCR1NPC1
SCHEMBL5657929 0.80 CXCR1 (0.51) CXCR2RAB9APOLBLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176310-B1 Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents UCB SA (GB) 2007-02-13 US claimed
US-7176310-B1 Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents UCB SA (GB) 2007-02-13 US disclosed