SCHEMBL56693

SCHEMBL56693

CS(=O)(=O)Nc1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 1.00
PGR P06401 1/20 0.67
NR3C2 P08235 5/20 0.64
CA1 P00915 2/20 0.58
CA2 P00918 2/20 0.58
PTGS2 P35354 2/20 0.58
HPGD P15428 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
ALDH1A1 P00352 2/20 0.58
KDM4E B2RXH2 1/20 0.58
LMNA P02545 1/20 0.58
HTT P42858 1/20 0.58
NPC1 O15118 1/20 0.56
AR P10275 1/20 0.56
RAB9A P51151 1/20 0.56
IL1RN P18510 1/20 0.56
ERAP1 Q9NZ08 1/20 0.56
CA12 O43570 1/20 0.56
CA9 Q16790 1/20 0.56
KDM1A O60341 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluoride SCHEMBL28258745 0.97 KEAP1 (0.95) KEAP1PGRNR3C2CA1CA2
Hydrogen Sulfide SCHEMBL27698561 0.97 KEAP1 (0.95) KEAP1PGRNR3C2CA1CA2
SCHEMBL11512295 0.97 KEAP1 (0.95) KEAP1PGRNR3C2CA1CA2
Hydrochloric Acid SCHEMBL27365433 0.97 KEAP1 (0.95) KEAP1PGRNR3C2CA1CA2
SCHEMBL1358244 0.91 KEAP1 (0.83) KEAP1PGRNR3C2CA1CA2
SCHEMBL9479898 0.91 KEAP1 (0.83) KEAP1PGRNR3C2CA1CA2
Boric Acid SCHEMBL6312485 0.91 KEAP1 (0.83) KEAP1PGRNR3C2CA1CA2
SCHEMBL27715693 0.87 KEAP1 (0.76) KEAP1PGRNR3C2CA1CA2
Ethyl Chloride SCHEMBL27421992 0.87 KEAP1 (0.76) KEAP1PGRNR3C2CA1CA2
SCHEMBL9387480 0.87 KEAP1 (0.76) KEAP1PGRNR3C2CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1575 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12004868-B2 Liposomal mitigation of drug-induced inhibition of the cardiac IKr channel SIGNPATH PHARMA INC. (US) 2024-06-11 US claimed
US-20230084927-A1 GLUCOSE UPTAKE INHIBITORS AND USES THEREOF METABOMED LTD. (IL) 2023-03-16 US claimed
CN-113200891-B Preparation method of cis-N-styryl amide derivative 华侨大学 2022-09-30 CN claimed
US-11279687-B2 Compounds and compositions for the inhibition of NAMPT VALO HEALTH, INC. (US) 2022-03-22 US claimed
CN-113200891-A Preparation method of cis-N-styryl amide derivative 华侨大学 2021-08-03 CN claimed
EP-3326616-B1 LIPOSOMAL MITIGATION OF DRUG-INDUCED LONG QT SYNDROME AND POTASSIUM DELAYED-RECTIFIER CURRENT SIGNPATH PHARMA INC (US) 2021-07-28 EP claimed
US-10617639-B2 Liposomal mitigation of drug-induced long QT syndrome and potassium delayed-rectifier current SIGNPATH PHARMA, INC. (US) 2020-04-14 US claimed
US-20200108056-A1 Liposomal Mitigation of Drug-Induced Inhibition of the Cardiac IKR Channel SIGNPATH PHARMA INC. 2020-04-09 US claimed
US-20190320975-A1 LIPOSOMAL MITIGATION OF DRUG-INDUCED INHIBITION OF THE CARDIAC IKR CHANNEL SIGNPATH PHARMA INC. 2019-10-24 US claimed
US-20190321293-A1 Liposomal Mitigation of Drug-Induced Long QT Syndrome and Potassium Delayed-Rectifier Current SIGNPATH PHARMA INC. 2019-10-24 US claimed
JP-2597176-B2 1997-04-02 JP claimed
EP-0441282-B1 Bichromophore methine and azamethine dyestuffs and a process for their transfer BASF AG (DE) 1993-12-15 EP claimed
EP-0441282-A1 Bichromophore methine and azamethine dyestuffs and a process for their transfer BASF Aktiengesellschaft (DE) 1991-08-14 EP claimed
US-4996284-A Heating a sulfonamide and epoxy resin in the presence of a Lewis Acid EMPAK, INC. 1991-02-26 US claimed
WO-1990013609-A1 NOVEL FLUORESCENT PIGMENT COMPOSITIONS AND A PROCESS FOR THEIR PREPARATION AND USE OF SAME MALLAVARAPU LEO X (US) 1990-11-15 WO claimed
WO-1990012829-A1 NOVEL EPOXY SULFONAMIDE-BASED RESINS, A PROCESS FOR THEIR PREPARATION AND USE OF SAME MALLAVARAPU LEO X (US) 1990-11-01 WO claimed
US-4929530-A OXIDATIVE LEUCO DYES, PHOTO-OXIDIZERS, REDUCING AGENTS, ORGANIC SULFONAMIDES AND PHENOLIC COMPONENTS; EXPOSING TO LIGHT FUJI PHOTO FILM CO., LTD. (JP) 1990-05-29 US claimed
CN-1038451-A Antiarrhythmics PFIZER LTD (GB) 1990-01-03 CN claimed
WO-1988005630-A1 FUNGICIDAL COMPOSITIONS SHELL AGRAR GMBH & CO. KG (DE) 1988-08-11 WO claimed
CN-87108295-A New alkane sulfonyl aniline derivative and its medicinal compositions and preparation method 1988-07-13 CN claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11279687-B2 Compounds and compositions for the inhibition of NAMPT NAMPT, NNT, NQO1 KEAP1 576/4885PGR 1495/4885NR3C2 1764/4885
US-20230084927-A1 GLUCOSE UPTAKE INHIBITORS AND USES THEREOF SLC2A4, SLC2A1, SLC2A2 KEAP1 199/4885PGR 2664/4885NR3C2 1252/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.