SCHEMBL5670577

SCHEMBL5670577

O=C1Nc2ccccc2OC1CCO

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.58
ALDH1A1 P00352 3/20 0.56
HPGD P15428 1/20 0.56
PARP1 P09874 1/20 0.54
GAA P10253 1/20 0.53
TP53 P04637 2/20 0.50
HSD17B10 Q99714 2/20 0.50
USP2 O75604 1/20 0.50
MAPK1 P28482 1/20 0.50
MAPT P10636 1/20 0.49
THRB P10828 1/20 0.49
TSHR P16473 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3641415 0.85 PARP1 (0.56) ALDH1A1HPGDPARP1GAATP53
SCHEMBL5671330 0.84 PARP1 (0.54) ALDH1A1HPGDPARP1GAATP53
SCHEMBL4821188 0.84 PARP1 (0.58) L3MBTL1ALDH1A1HPGDPARP1GAA
SCHEMBL7471863 0.82 L3MBTL1 (0.59) L3MBTL1ALDH1A1HPGDPARP1GAA
SCHEMBL9155928 0.81 PARP1 (0.51) ALDH1A1HPGDPARP1GAATP53
SCHEMBL5670690 0.81 PARP1 (0.55) ALDH1A1HPGDPARP1GAATP53
SCHEMBL5671346 0.81 ALDH1A1 (0.54) ALDH1A1HPGDPARP1GAATP53
SCHEMBL22186873 0.81 PARP1 (0.51) ALDH1A1HPGDPARP1GAATP53
SCHEMBL5672408 0.81 ALDH1A1 (0.40) L3MBTL1ALDH1A1HPGDPARP1GAA
SCHEMBL5671433 0.80 BRD4 (0.55) ALDH1A1HPGDPARP1GAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023180189-A1 MPRO TARGETING ANTIVIRAL COMPOUNDS EXSCIENTIA AI LIMITED (GB) 2023-09-28 WO disclosed
EP-0980362-B1 SUBSTITUTED HETEROCYCLES AND THEIR USE IN MEDICAMENTS SCHERING AG (DE) 2006-08-16 EP disclosed
EP-0869949-B1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO MCNEIL PHARM INC (US) 2002-12-18 EP disclosed
US-6191127-B1 ANTIINFLAMMATORY AGENTS, AUTOIMMUNE DISEASES, CARDIOVASCULAR DISORDERS, NERVOUS SYSTEM DISORDERS SCHERING AKTIENGESELLSCHAFT (DE) 2001-02-20 US disclosed
EP-0980362-A1 SUBSTITUTED HETEROCYCLES AND THEIR USE IN MEDICAMENTS SCHERING AKTIENGESELLSCHAFT (DE) 2000-02-23 EP disclosed
US-5854242-A Benzoxazine antimicrobial agents ORTHO PHARMACEUTICAL CORPORATION (US) 1998-12-29 US disclosed
WO-1998050372-A1 SUBSTITUTED HETEROCYCLES AND THEIR USE IN MEDICAMENTS SCHERING AKTIENGESELLSCHAFT (DE) 1998-11-12 WO disclosed
EP-0869949-A1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1998-10-14 EP disclosed
US-5696117-A BACTERICIDE ORTHO PHARMACEUTICAL CORPORATION (US) 1997-12-09 US disclosed
WO-1997017333-A1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1997-05-15 WO disclosed