SCHEMBL5682140

SCHEMBL5682140

C=C(C(=O)OCc1ccccc1)C(CC(C)C)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSB P07858 2/20 0.49
ALDH1A1 P00352 3/20 0.47
CTSK P43235 5/20 0.47
CTSS P25774 2/20 0.44
CTSL P07711 1/20 0.44
SLC15A1 P46059 1/20 0.44
CAPN1 P07384 1/20 0.44
ACE2 Q9BYF1 1/20 0.43
MAPK1 P28482 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A3 Q01959 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5682142 1.00 CTSB (0.49) CTSBALDH1A1CTSKCTSSCTSL
SCHEMBL5680064 0.87 CTSK (0.44) CTSBALDH1A1CTSKCTSSCTSL
SCHEMBL5680067 0.87 CTSK (0.44) CTSBALDH1A1CTSKCTSSCTSL
SCHEMBL9507442 0.83 ALDH1A1 (0.47) ALDH1A1SLC15A1MAPK1L3MBTL1SLC6A2
SCHEMBL16681232 0.83 CTSB (0.61) CTSBALDH1A1CTSKCTSSCTSL
SCHEMBL7279716 0.83 ALDH1A1 (0.55) ALDH1A1CTSKSLC15A1MAPK1L3MBTL1
SCHEMBL11707070 0.83 CTSB (0.61) CTSBALDH1A1CTSKCTSSCTSL
SCHEMBL5678072 0.83 CACNA1B (0.44) CTSKCTSSCTSL
SCHEMBL5677963 0.83 CACNA1B (0.44) CTSKCTSSCTSL
Hydrochloric Acid SCHEMBL11707065 0.81 CTSB (0.60) CTSBALDH1A1CTSKCTSSCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934292-B1 METALLOPROTEINASE INHIBITORS VERNALIS OXFORD LTD (GB) 2006-03-15 EP disclosed
EP-1066273-A1 METALLOPROTEINASE INHIBITORS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 2001-01-10 EP disclosed
US-6022873-A Metalloproteinase inhibitors BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 2000-02-08 US disclosed
WO-1999048881-A1 METALLOPROTEINASE INHIBITORS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1999-09-30 WO disclosed
EP-0934292-A1 METALLOPROTEINASE INHIBITORS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1999-08-11 EP disclosed
WO-1998017655-A1 METALLOPROTEINASE INHIBITORS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1998-04-30 WO disclosed