SCHEMBL5686228

SCHEMBL5686228

COc1cc(OC)cc(N2CCCNCC2)c1

nearest known ligand 0.86

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 3/20 0.86
CHRNB2 P17787 6/20 0.70
CHRNA4 P43681 6/20 0.70
HTR3A P46098 4/20 0.64
HTR3E A5X5Y0 2/20 0.64
HTR3B O95264 2/20 0.64
HTR3D Q70Z44 2/20 0.64
HTR3C Q8WXA8 2/20 0.64
SIGMAR1 Q99720 1/20 0.64
HTR1A P08908 3/20 0.56
HTR1D P28221 2/20 0.56
HTR1B P28222 1/20 0.56
TGFBR1 P36897 1/20 0.56
HTR7 P34969 2/20 0.53
HTR2B P41595 2/20 0.53
ACVR1 Q04771 1/20 0.52
HTR2C P28335 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL443521 0.93 ADRB1 (1.00) ADRB1CHRNB2CHRNA4HTR3AHTR3E
Hydrochloric Acid SCHEMBL18577062 0.91 ADRB1 (0.96) ADRB1CHRNB2CHRNA4HTR3AHTR3E
SCHEMBL5237992 0.86 ADRB1 (0.86) ADRB1CHRNB2CHRNA4HTR3AHTR3E
SCHEMBL4526848 0.85 ADRB1 (0.88) ADRB1CHRNB2CHRNA4HTR3AHTR3E
SCHEMBL5664269 0.83 CHRNB2 (1.00) ADRB1CHRNB2CHRNA4
SCHEMBL2873315 0.83 ADRB1 (0.80) ADRB1CHRNB2CHRNA4HTR3AHTR3E
SCHEMBL4925469 0.81 ADRB1 (0.77) ADRB1CHRNB2CHRNA4HTR3AHTR3E
SCHEMBL8891314 0.81 ADRB1 (0.77) ADRB1CHRNB2CHRNA4HTR3AHTR3E
SCHEMBL5682967 0.81 ADRB1 (0.77) ADRB1CHRNB2CHRNA4HTR3AHTR3E
SCHEMBL11922738 0.81 ADRB1 (0.66) ADRB1CHRNB2CHRNA4HTR3AHTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1645556-A1 Arylpiperazine-benzoylamide derivatives useful as pharmaceutical agents Boehringer Ingelheim International GmbH (DE) 2006-04-12 EP disclosed